SCHEMBL9434017

SCHEMBL9434017

COc1cccc2sc(C(N)=O)c(N(C)C)c12

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
STING1 Q86WV6 2/20 0.46
IKBKB O14920 4/20 0.42
SLC9A1 P19634 2/20 0.40
BACE1 P56817 1/20 0.40
ALDH1A1 P00352 2/20 0.40
GAA P10253 1/20 0.40
HPGD P15428 1/20 0.40
HSD17B10 Q99714 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
KMT2A Q03164 2/20 0.39
PRNP P04156 1/20 0.38
TSHR P16473 1/20 0.38
MAPK1 P28482 1/20 0.38
PPARG P37231 1/20 0.38
HTT P42858 1/20 0.38
MAPK10 P53779 1/20 0.38
NCOA2 Q15596 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
RXFP1 Q9HBX9 1/20 0.38
HDAC3 O15379 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9433956 0.86 BACE1 (0.48) STING1BACE1ALDH1A1GAAHPGD
SCHEMBL9433877 0.81 IKBKB (0.58) STING1IKBKBSLC9A1BACE1ALDH1A1
SCHEMBL9434315 0.80 MAPK1 (0.51) STING1IKBKBALDH1A1HPGDL3MBTL1
SCHEMBL7218005 0.71 KDM4E (0.60) STING1IKBKBBACE1ALDH1A1GAA
SCHEMBL26049804 0.71 EDNRA (0.50) STING1BACE1ALDH1A1GAAHPGD
SCHEMBL11101251 0.70 BACE1 (0.54) BACE1ALDH1A1GAAHPGDHSD17B10
SCHEMBL9434117 0.69 ALDH1A1 (0.49) STING1ALDH1A1GAAHPGDHSD17B10
SCHEMBL22908903 0.68 STING1 (0.47) STING1BACE1MAPK1HDAC3HDAC4
SCHEMBL9024186 0.68 STING1 (0.42) STING1IKBKBSLC9A1ALDH1A1GAA
SCHEMBL1030218 0.68 CA12 (0.65) ALDH1A1HPGDHSD17B10L3MBTL1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5350748-A 3-thio or amino substituted-benzo[b]thiophene-2-carboxamides and 3-oxygen, thio, or amino substituted-benzofuran-2-carboxamides as inhibitors of cell adhesion WARNER-LAMBERT COMPANY (US) 1994-09-27 US disclosed