SCHEMBL9434216

SCHEMBL9434216

COC(=O)C1=C(C)NC(C)=C(c2ccccn2)C1c1cccc(I)c1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 3/20 0.58
KDM4E B2RXH2 3/20 0.58
CACNA1B Q00975 2/20 0.47
CASP1 P29466 2/20 0.46
CASP7 P55210 1/20 0.46
ADORA3 P0DMS8 1/20 0.46
ALDH1A1 P00352 1/20 0.46
GAA P10253 1/20 0.46
HPGD P15428 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
HIF1A Q16665 3/20 0.43
MEN1 O00255 2/20 0.43
CYP1A2 P05177 2/20 0.43
CYP3A4 P08684 2/20 0.43
CYP2C9 P11712 2/20 0.43
CYP2C19 P33261 2/20 0.43
KMT2A Q03164 2/20 0.43
MAPT P10636 2/20 0.43
CACNA1F O60840 2/20 0.43
CACNA1D Q01668 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10432260 0.89 HSD17B10 (0.60) HSD17B10KDM4ECACNA1BCASP1CASP7
SCHEMBL9434036 0.88 CACNA1B (0.52) HSD17B10KDM4ECACNA1BCASP1
SCHEMBL9433668 0.88 HSD17B10 (0.61) HSD17B10KDM4ECACNA1BCASP1CASP7
SCHEMBL9434200 0.88 KDM4E (0.58) HSD17B10KDM4ECASP1CASP7ADORA3
SCHEMBL9434198 0.88 HSD17B10 (0.58) HSD17B10KDM4ECACNA1BCASP1CASP7
SCHEMBL9433631 0.88 HSD17B10 (0.58) HSD17B10KDM4ECACNA1BCASP1CASP7
SCHEMBL9433755 0.85 CACNA1F (0.60) HSD17B10KDM4ECACNA1BCASP1CASP7
SCHEMBL9434383 0.84 MAPT (0.64) ADORA3SMN1; SMN2HIF1AMEN1CYP1A2
SCHEMBL9434343 0.84 KDM4E (0.64) HSD17B10KDM4ECACNA1BCASP1CASP7
SCHEMBL9434370 0.83 KDM4E (0.60) HSD17B10KDM4ECACNA1BCASP1CASP7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5276150-A Vasodilators, anticoagulants, calcium channel blockers FUJIREBIO INC. (JP) 1994-01-04 US disclosed
EP-0400660-A1 1,4-dihydropyridine derivatives FUJIREBIO INC. (JP) 1990-12-05 EP disclosed