SCHEMBL9434302

SCHEMBL9434302

COc1ccc2c(c1)CCN(CC#N)C2C

nearest known ligand 0.47

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
DRD1 P21728 4/20 0.47
CA1 P00915 4/20 0.45
CA2 P00918 4/20 0.45
CA9 Q16790 4/20 0.45
CA14 Q9ULX7 4/20 0.45
DRD2 P14416 3/20 0.44
DRD4 P21917 2/20 0.44
DRD5 P21918 2/20 0.44
DRD3 P35462 2/20 0.44
PRMT5 O14744 1/20 0.43
HTR2C P28335 1/20 0.43
S1PR1 P21453 1/20 0.41
SIGMAR1 Q99720 1/20 0.41
KDM4E B2RXH2 1/20 0.40
KMT2A Q03164 1/20 0.40
ADRA1A P35348 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9433750 0.80 DRD1 (0.48) DRD1CA1CA2CA9CA14
SCHEMBL28239143 0.79 DRD1 (0.50) DRD1CA1CA2CA9CA14
SCHEMBL8024197 0.76 MAOA (0.60) DRD1CA1CA2CA9CA14
SCHEMBL4764318 0.74 DRD1 (0.51) DRD1CA1CA2CA9CA14
SCHEMBL10659360 0.74 CA1 (0.49) DRD1CA1CA2CA9CA14
Hydrochloric Acid SCHEMBL10663782 0.73 CA1 (0.48) DRD1CA1CA2CA9CA14
SCHEMBL10663768 0.72 HRH3 (0.44) DRD1DRD2DRD4DRD5DRD3
SCHEMBL5518952 0.72 DRD1 (0.51) DRD1CA1CA2CA9CA14
SCHEMBL10662717 0.72 HRH3 (0.41) DRD1DRD2DRD4PRMT5HTR2C
Hydrochloric Acid SCHEMBL10659895 0.72 HRH3 (0.44) DRD1DRD2DRD4SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5294621-A Thieno tetrahydropyridines useful as class III antiarrhythmic agents ORTHO PHARMACEUTICAL CORPORATION (US) 1994-03-15 US disclosed