SCHEMBL9434307

SCHEMBL9434307

[CH2]/C=C/C#Cc1ccccc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
APP P05067 1/20 0.50
MAPT P10636 5/20 0.39
CYP3A4 P08684 3/20 0.38
CYP1A2 P05177 2/20 0.38
CYP2C9 P11712 2/20 0.38
CYP2C19 P33261 2/20 0.38
THPO P40225 1/20 0.38
BLM P54132 1/20 0.37
PMP22 Q01453 1/20 0.37
GRM5 P41594 1/20 0.37
HCAR2 Q8TDS4 1/20 0.36
ALDH1A1 P00352 3/20 0.36
MEN1 O00255 2/20 0.36
HPGD P15428 2/20 0.36
KMT2A Q03164 2/20 0.36
USP2 O75604 1/20 0.36
PLA2G1B P04054 1/20 0.36
ATG4B Q9Y4P1 1/20 0.36
NPC1 O15118 2/20 0.35
KDM4E B2RXH2 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5507856 0.85 APP (0.61) APPMAPTCYP3A4CYP1A2CYP2C9
SCHEMBL5507858 0.85 APP (0.61) APPMAPTCYP3A4CYP1A2CYP2C9
SCHEMBL9146168 0.85 APP (0.61) APPMAPTCYP3A4CYP1A2CYP2C9
SCHEMBL28978993 0.77 APP (0.46) APPMAPTCYP3A4CYP1A2CYP2C9
SCHEMBL5100967 0.76 APP (0.50) APPMAPTCYP3A4CYP1A2CYP2C9
SCHEMBL5100970 0.76 APP (0.50) APPMAPTCYP3A4CYP1A2CYP2C9
SCHEMBL136424 0.75 APP (0.55) APPMAPTCYP3A4CYP1A2CYP2C9
SCHEMBL840229 0.75 APP (0.55) APPMAPTCYP3A4CYP1A2CYP2C9
SCHEMBL3888887 0.74 APP (0.48) APPMAPTCYP3A4CYP1A2CYP2C9
SCHEMBL3888883 0.74 APP (0.48) APPMAPTCYP3A4CYP1A2CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5276150-A Vasodilators, anticoagulants, calcium channel blockers FUJIREBIO INC. (JP) 1994-01-04 US claimed
EP-0400660-A1 1,4-dihydropyridine derivatives FUJIREBIO INC. (JP) 1990-12-05 EP claimed
US-5276150-A Vasodilators, anticoagulants, calcium channel blockers FUJIREBIO INC. (JP) 1994-01-04 US disclosed