SCHEMBL9434812

SCHEMBL9434812

CCCCCOC(=O)/C=C(/C)N

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCAR2 Q8TDS4 3/20 0.55
ATM Q13315 1/20 0.53
TSHR P16473 5/20 0.50
HPGD P15428 1/20 0.50
NPSR1 Q6W5P4 2/20 0.49
MAPT P10636 1/20 0.49
RAB9A P51151 1/20 0.49
NAAA Q02083 1/20 0.47
ALDH1A1 P00352 2/20 0.47
EPHX1 P07099 1/20 0.44
HTR2C P28335 1/20 0.42
PRSS1 P07477 1/20 0.41
PRSS2 P07478 1/20 0.41
PRSS3 P35030 1/20 0.41
CES2 O00748 1/20 0.41
APP P05067 1/20 0.41
CYP3A4 P08684 2/20 0.41
TP53 P04637 1/20 0.41
MAPK1 P28482 1/20 0.41
RAD52 P43351 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7430462 1.00 HCAR2 (0.55) HCAR2ATMTSHRHPGDNPSR1
SCHEMBL9434472 0.98 HCAR2 (0.56) HCAR2ATMTSHRHPGDNPSR1
SCHEMBL9434488 0.98 HCAR2 (0.56) HCAR2ATMTSHRHPGDNPSR1
SCHEMBL10543217 0.98 HCAR2 (0.56) HCAR2ATMTSHRHPGDNPSR1
SCHEMBL10902247 0.98 HCAR2 (0.56) HCAR2ATMTSHRHPGDNPSR1
SCHEMBL9433613 0.98 HCAR2 (0.56) HCAR2ATMTSHRHPGDNPSR1
SCHEMBL10898563 0.98 HCAR2 (0.56) HCAR2ATMTSHRHPGDNPSR1
SCHEMBL10925831 0.98 HCAR2 (0.56) HCAR2ATMTSHRHPGDNPSR1
SCHEMBL9433770 0.98 HCAR2 (0.56) HCAR2ATMTSHRHPGDNPSR1
SCHEMBL10902234 0.98 HCAR2 (0.56) HCAR2ATMTSHRHPGDNPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5276150-A Vasodilators, anticoagulants, calcium channel blockers FUJIREBIO INC. (JP) 1994-01-04 US disclosed
EP-0400660-A1 1,4-dihydropyridine derivatives FUJIREBIO INC. (JP) 1990-12-05 EP disclosed
EP-0225574-B1 NOVEL 1,4-DIHYDROPYRIDINES CONTAINING FLUORINE, PROCESS FOR THEIR PREPARATION AND THEIR USE AS MEDICAMENTS BAYER AG (DE) 1990-05-16 EP disclosed
US-4874773-A HYPOTENSIVE AGENTS, VASODILATORS NIPPON SHOJI KABUSHIKI KAISHA (JP) 1989-10-17 US disclosed
US-4798840-A Coronary-active fluorine-containing 1,4-dihydropyridines BAYER AKTIENGESELLSCHAFT (DE) 1989-01-17 US disclosed
EP-0225574-A1 Novel 1,4-dihydropyridines containing fluorine, process for their preparation and their use as medicaments BAYER AG (DE) 1987-06-16 EP disclosed
EP-0220653-A2 3-Aminocarbonyl-1,4-dihydropyridine-5-carboxylic acid compounds, process for preparation and use thereof, and pharmaceutical composition containing the same Nippon Shoji Kabushiki Kaisha (JP) 1987-05-06 EP disclosed