SCHEMBL943489

SCHEMBL943489

COc1cccc(-c2cccc(C3(C4CCOCC4)N=C(C)C(N)=N3)c2)c1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 20/20 1.00
KCNH2 Q12809 11/20 1.00
BACE2 Q9Y5Z0 3/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL946784 0.87 BACE1 (0.76) BACE1KCNH2BACE2
SCHEMBL1075789 0.85 BACE1 (0.74) BACE1KCNH2BACE2
SCHEMBL6891914 0.83 BACE1 (0.71) BACE1KCNH2BACE2
SCHEMBL932637 0.82 BACE1 (0.86) BACE1KCNH2BACE2
SCHEMBL932037 0.81 BACE1 (0.68) BACE1KCNH2BACE2
SCHEMBL932138 0.74 BACE1 (1.00) BACE1KCNH2
SCHEMBL6893840 0.74 BACE1 (1.00) BACE1KCNH2
SCHEMBL1075786 0.74 BACE1 (0.58) BACE1KCNH2BACE2
SCHEMBL932718 0.73 BACE1 (0.58) BACE1KCNH2BACE2
SCHEMBL6892665 0.73 BACE1 (0.80) BACE1KCNH2BACE2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011002408-A1 NOVEL COMPOUNDS FOR TREATMENT OF NEURODEGENERATION ASSOCIATED WITH DISEASES, SUCH AS ALZHEIMER'S DISEASE OR DEMENTIA ASTRAZENECA AB (SE) 2011-01-06 WO disclosed