SCHEMBL9435338

SCHEMBL9435338

Cc1cccc(NC(=O)NC2CSc3ccccc3N(CC(=O)N3CCC4(CC3)OCCO4)C2=O)c1

nearest known ligand 0.58

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CCKBR P32239 15/20 0.58
ALDH1A1 P00352 2/20 0.44
CYP1A2 P05177 1/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2C19 P33261 1/20 0.44
MAPT P10636 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8904425 0.89 CCKBR (0.61) CCKBRALDH1A1MAPT
SCHEMBL8903356 0.89 CCKBR (0.60) CCKBR
SCHEMBL8903101 0.85 CCKBR (0.60) CCKBR
SCHEMBL8904274 0.85 CCKBR (0.60) CCKBRALDH1A1MAPT
SCHEMBL8904296 0.85 CCKBR (0.60) CCKBR
SCHEMBL8903106 0.85 CCKBR (0.60) CCKBR
SCHEMBL8904532 0.85 CCKBR (0.62) CCKBR
SCHEMBL9435384 0.85 CCKBR (0.60) CCKBR
SCHEMBL8905032 0.83 CCKBR (0.57) CCKBRALDH1A1MAPT
SCHEMBL8905038 0.83 CCKBR (0.57) CCKBRALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1994001421-A1 BENZOTHIAZEPINE AND BENZOXAZEPINE DERIVATIVES AS CHOLECYSTOKININ RECEPTOR ANTAGONISTS PFIZER INC. (US) 1994-01-20 WO disclosed