SCHEMBL9435548

SCHEMBL9435548

COCc1nc[nH]c1C

nearest known ligand 0.00

⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL11198159 0.98 TDP1 (0.55)
SCHEMBL11379774 0.79 HRH2 (0.50)
SCHEMBL11381375 0.76 HRH2 (0.47)
SCHEMBL2830891 0.75
SCHEMBL9624460 0.74 GABRR1 (0.54)
SCHEMBL2830017 0.74 HRH2 (0.44)
SCHEMBL4905447 0.73
SCHEMBL5791428 0.73
SCHEMBL8014968 0.73
SCHEMBL10376001 0.73

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0279161-B1 A process for the preparation of cimetidine LEK TOVARNA FARMACEVTSKIH (SI) 1994-01-05 EP disclosed
US-4855439-A Process for the preparation of cimetidine LEK (YU) 1989-08-08 US disclosed
EP-0279161-A2 A process for the preparation of cimetidine LEK, tovarna farmacevtskih in kemicnih izdelkov, n.sol.o. (SI) 1988-08-24 EP disclosed
US-4267337-A Imidazolemethylphosphonium salts SK&F LAB CO. (US) 1981-05-12 US disclosed
US-4215217-A Process for preparing 4-substituted imidazole compounds SK&F LAB CO. (US) 1980-07-29 US disclosed
US-4200761-A Process for preparing N-cyano-N'methyl-N\"-{2-[(4-methyl-5-imidazolyl)-methylthio]-ethyl} guanidine LEK, TOVARNA FARMACEVTSKIH IN KEMICNIH IZDELKOV, N.SOL.O. (YU) 1980-04-29 US disclosed
US-4163858-A Process for preparing new imidazolemethylphosphonium salts SK&F LAB CO. (US) 1979-08-07 US disclosed
US-4139708-A Intermediates and processes useful for preparing medicinal agents imidazolemethylphosphonium salts SK&F LAB CO. (US) 1979-02-13 US disclosed
US-4119781-A Process for preparing 4-substituted imidazole compounds SK&F LAB CO. (US) 1978-10-10 US disclosed
US-4104472-A Imidazolemethylphosphonium salts SMITHKLINE CORPORATION (US) 1978-08-01 US disclosed