SCHEMBL943759

SCHEMBL943759

Cc1cc(N)c(Cl)cc1Cl

nearest known ligand 0.75

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CD44 P16070 1/20 0.75
GAA P10253 1/20 0.58
NPC1 O15118 1/20 0.50
CYP3A4 P08684 7/20 0.48
TSHR P16473 5/20 0.46
MAPK1 P28482 2/20 0.46
TP53 P04637 1/20 0.40
ALDH1A1 P00352 5/20 0.39
GRIN2D O15399 1/20 0.38
GRIN3B O60391 1/20 0.38
GRIN1 Q05586 1/20 0.38
GRIN2A Q12879 1/20 0.38
GRIN2B Q13224 1/20 0.38
GRIN2C Q14957 1/20 0.38
GRIN3A Q8TCU5 1/20 0.38
CA12 O43570 1/20 0.37
CA1 P00915 1/20 0.37
CA2 P00918 1/20 0.37
CA7 P43166 1/20 0.37
CA9 Q16790 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8341703 0.89 CD44 (0.75) CD44GAANPC1CYP3A4TSHR
SCHEMBL16282614 0.86 CD44 (0.62) CD44GAANPC1CYP3A4TSHR
SCHEMBL404439 0.86 CD44 (1.00) CD44GAANPC1CYP3A4TSHR
SCHEMBL11826575 0.85 CD44 (0.56) CD44GAANPC1CYP3A4TSHR
SCHEMBL203360 0.83 CD44 (0.75) CD44GAANPC1CYP3A4TSHR
SCHEMBL29683620 0.83 GAA (0.67) CD44GAANPC1CYP3A4TSHR
SCHEMBL2026149 0.83 GAA (0.67) CD44GAANPC1CYP3A4TSHR
Hydrochloric Acid SCHEMBL7676240 0.83 CD44 (0.94) CD44GAACYP3A4TSHRMAPK1
SCHEMBL9069642 0.81 CD44 (0.56) CD44GAANPC1CYP3A4TSHR
Hydrochloric Acid SCHEMBL8647124 0.81 CD44 (0.64) CD44GAANPC1CYP3A4TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 93 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0653412-B1 Process for preparing 4,5-difluorobenzaldehydes BAYER AG (DE) 1998-01-21 EP claimed
US-5489715-A Process for preparing 4,5-difluorobenzaldehydes BAYER AKTIENGESELLSCHAFT (DE) 1996-02-06 US claimed
EP-0653412-A1 Process for preparing 4,5-difluorobenzaldehydes BAYER AG (DE) 1995-05-17 EP claimed
EP-0077501-B1 PROCESS FOR THE PREPARATION OF FLUOROAROMATIC COMPOUNDS SUBSTITUTED IN THE ORTHO POSITION BAYER AG (DE) 1985-05-22 EP claimed
US-4476320-A REACTION OF AN ANILINE TO FORM DIAZONIUM TETRAFLUOROBORATE, DECOMPOSITION BAYER AKTIENGESELLSCHAFT (DE) 1984-10-09 US claimed
US-4439620-A CHEMICAL INTERMEDIATE BAYER AKTIENGESELLSCHAFT (DE) 1984-03-27 US claimed
EP-0077501-A1 Process for the preparation of fluoroaromatic compounds substituted in the ortho position BAYER AG (DE) 1983-04-27 EP claimed
CN-119255992-A Heterocyclic derivatives, compositions and uses thereof 北京丹擎医药科技有限公司 2025-01-03 CN disclosed
WO-2023226964-A1 HETEROCYCLIC DERIVATIVES, COMPOSITIONS AND USES THEREOF DANATLAS PHARMACEUTICALS CO., LTD. (CN) 2023-11-30 WO disclosed
EP-4001269-A1 BENZOISOTHIAZOLE, ISOTHIAZOLO[3,4-B]PYRIDINE, QUINAZOLINE, PHTHALAZINE, PYRIDO[2,3-D]PYRIDAZINE AND PYRIDO[2,3-D]PYRIMIDINE DERIVATIVES AS KRAS G12C INHIBITORS FOR TREATING LUNG, PANCREATIC OR COLORECTAL CANCER Amgen Inc. (US) 2022-05-25 EP disclosed
WO-2021219090-A1 QUINOXALINE DIONE DERIVATIVE AS IRREVERSIBLE INHIBITOR OF KRAS G12C MUTANT PROTEIN 北京泰德制药股份有限公司 (CN) 2021-11-04 WO disclosed
WO-2021202600-A1 SMALL MOLECULE INHIBITORS OF INFLUENZA HEMAGGLUTININ THE SCRIPPS RESEARCH INSTITUTE (US) 2021-10-07 WO disclosed
US-9580444-B2 Polycyclic pyrazolinone derivative and herbicide comprising same as effective component thereof SAGAMI CHEMICAL RESEARCH INSTITUTE (JP) 2017-02-28 US disclosed
US-4038268-A DIAZOTIZATION, COUPLING BAYER AKTIENGESELLSCHAFT (DT) 1977-07-26 US disclosed
US-4006128-A CELLULOSE ACETATES, VINYL POLYMERS, POLYOLEFINS, POLYESTERS BAYER AKTIENGESELLSCHAFT (DT) 1977-02-01 US disclosed
US-3975534-A Pharmaceutical compositions useful for treating tick infestation in animals which contain 2-aryliminopyrrolidines or their salts as the active agent BAYER AKTIENGESELLSCHAFT (DT) 1976-08-17 US disclosed
US-3962209-A PROCESS FOR PREPARING AZO DYESTUFFS WITH ORTHO-AZO CYANO GROUPS BY CYANO EXCHANGE OF METAL CYANIDES AND HALO DYESTUFFS BAYER AKTIENGESELLSCHAFT (DT) 1976-06-08 US disclosed
US-3957749-A WATER-INSOLUBLE MONOAZO PYRIDINE DYES CASSELLA FARBWERKE MAINKUR AKTIENGESELLSCHAFT (DT) 1976-05-18 US disclosed
US-3956264-A Basic azo dyestuffs having indolyl-methyleneamino substituent in the diazo component BAYER AKTIENGESELLSCHAFT (DT) 1976-05-11 US disclosed
US-3953420-A Azo pigments derived from 2-hydroxy-3-carboxynaphthalene containing a substituted or unsubstituted phthalimide BADISCHE ANILIN- & SODA-FABRIK AKTIENGESELLSCHAFT (DT) 1976-04-27 US disclosed