SCHEMBL9446263

SCHEMBL9446263

c1ccc(N(Cc2cccc3ccccc23)c2ccccc2)cc1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 4/20 0.60
CYP2C19 P33261 3/20 0.60
CYP2D6 P10635 3/20 0.60
TDP1 Q9NUW8 1/20 0.48
CYP2C9 P11712 1/20 0.48
LMNA P02545 3/20 0.47
NR1I2 O75469 2/20 0.47
SLC6A2 P23975 2/20 0.47
HTR2A P28223 2/20 0.47
SLC6A4 P31645 2/20 0.47
KCNH2 Q12809 2/20 0.47
SIGMAR1 Q99720 2/20 0.47
MEN1 O00255 2/20 0.47
KMT2A Q03164 2/20 0.47
HTT P42858 2/20 0.47
DRD2 P14416 1/20 0.47
ADRA2C P18825 1/20 0.47
CNR1 P21554 1/20 0.47
ADRA1A P35348 1/20 0.47
OPRK1 P41145 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9446248 0.89 CYP1A2 (0.53) CYP1A2CYP2C19CYP2D6TDP1CYP2C9
SCHEMBL9446285 0.86 CYP2D6 (0.62) CYP1A2CYP2C19CYP2D6TDP1CYP2C9
SCHEMBL9446227 0.86 L3MBTL1 (0.51) CYP1A2CYP2C19CYP2D6TDP1NR1I2
SCHEMBL5362452 0.81 CYP2D6 (0.67) CYP1A2CYP2C19CYP2D6TDP1CYP2C9
SCHEMBL18784910 0.79 KMT2A (0.46) CYP1A2CYP2C19CYP2D6TDP1CYP2C9
SCHEMBL7915221 0.79 CYP2D6 (0.69) CYP1A2CYP2C19CYP2D6TDP1CYP2C9
SCHEMBL6678833 0.78 CYP2D6 (0.53) CYP1A2CYP2C19CYP2D6TDP1CYP2C9
SCHEMBL820553 0.75 CYP2D6 (0.77) CYP1A2CYP2C19CYP2D6TDP1CYP2C9
SCHEMBL10932466 0.75 CYP2D6 (1.00) CYP1A2CYP2C19CYP2D6CYP2C9LMNA
SCHEMBL31316173 0.75 CYP2D6 (0.77) CYP1A2CYP2C19CYP2D6TDP1CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5196606-A Aromatic tertiary amines, enamines, deoxybenzoins and benzils HAY ALLAN S (CA) 1993-03-23 US disclosed
US-5117062-A Aromatic tertiary amines, enamines, deoxybenzoins and benzils HAY ALLAN S (CA) 1992-05-26 US disclosed
US-5011998-A Aromatic tertiary amines, enamines, deoxybenzoins and benzils HAY ALLAN S (CA) 1991-04-30 US disclosed