Pnu-82965

Pnu-82965

SCHEMBL9447616

CC(=O)NCC1CN(c2ccc3c(c2)CCC3=O)C(=O)O1

nearest known ligand 0.60

Full drug profile on Sugi Atlas →

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
MAOA P21397 5/20 0.59
MAOB P27338 2/20 0.57
PTGS1 P23219 2/20 0.57
SDHA P31040 2/20 0.57
LMNA P02545 1/20 0.57
CALML3 P27482 1/20 0.57
F10 P00742 5/20 0.48
ABCB11 O95342 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Pnu-82965 SCHEMBL9447627 1.00 MAOA (0.59) MAOAMAOBPTGS1SDHALMNA
SCHEMBL9447577 0.94 MAOA (0.57) MAOAMAOBPTGS1SDHALMNA
SCHEMBL9447588 0.94 MAOA (0.57) MAOAMAOBPTGS1SDHALMNA
SCHEMBL6191933 0.94 MAOA (0.57) MAOAMAOBPTGS1SDHALMNA
SCHEMBL6194275 0.94 MAOA (0.57) MAOAMAOBPTGS1SDHALMNA
SCHEMBL6238447 0.88 MAOA (0.58) MAOAMAOBPTGS1SDHALMNA
SCHEMBL6236130 0.88 MAOA (0.58) MAOAMAOBPTGS1SDHALMNA
SCHEMBL6236134 0.88 MAOA (0.58) MAOAMAOBPTGS1SDHALMNA
SCHEMBL6238455 0.88 MAOA (0.58) MAOAMAOBPTGS1SDHALMNA
SCHEMBL6235269 0.87 MAOA (0.64) MAOAMAOBPTGS1SDHALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 22 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0311090-A1 Aminomethyl oxooxazolidinyl cycloalkylbenzene derivatives useful as antibacterial agents THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1989-04-12 EP claimed
US-4801600-A Aminomethyl oxooxazolidinyl cycloalkylbenzene derivatives useful as antibacterial agents E. I. DU PONT DE NEMOURS AND COMPANY (US) 1989-01-31 US claimed
US-5225565-A Antibacterial 3-(fused-ring substituted)phenyl-5β-amidomethyloxazolidin-2-ones THE UPJOHN COMPANY (US) 1993-07-06 US disclosed
US-5182403-A Bactericides, treatment of AIDS THE UPJOHN COMPANY (US) 1993-01-26 US disclosed
US-5164510-A Bactericides THE UPJOHN COMPANY (US) 1992-11-17 US disclosed
US-5039690-A Aminomethyl oxooxazolidinyl oxa or thia cycloalkylbenzene derivatives useful as antibacterial agents DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1991-08-13 US disclosed
US-5036093-A Effective against grampositive bacteria including some antibiotic resistant strains DU PONT MERCK PHARMACEUTICAL (US) 1991-07-30 US disclosed
US-5036092-A Effective against antibiotic resistant streptococci and staphylococci DU PONT MERCK PHARMACEUTICAL (US) 1991-07-30 US disclosed
US-5032605-A Aminomethyl oxooxazolidinyl oxa or thia cycloalkylbenzene derivatives useful as antibacterial agents DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1991-07-16 US disclosed
EP-0434714-A1 IN POSITION 3 SUBSTITUTED-5-BETA-AMIDOMETHYL-OXAZOLIDIN-2-ONES THE UPJOHN COMPANY (US) 1991-07-03 EP disclosed
US-4985429-A Aminomethyl oxooxazolidinyl cycloalkylbenzene derivatives useful as antibacterial agents E. I. DU PONT DE NEMOURS AND COMPANY (US) 1991-01-15 US disclosed
US-4965268-A ADMINISTERING TO A BACTERIAL INFECTION IN A MAMMAL E. I. DU PONT DE NEMOURS AND COMPANY (US) 1990-10-23 US disclosed
US-4921869-A Aminomethyl oxooxazolidinyl cycloalkylbenzene derivatives useful as antibacterial agents E. I. DU PONT DE NEMOURS AND COMPANY (US) 1990-05-01 US disclosed
US-4921869-A Aminomethyl oxooxazolidinyl cycloalkylbenzene derivatives useful as antibacterial agents E. I. DU PONT DE NEMOURS AND COMPANY (US) 1990-05-01 US disclosed
WO-1990002744-A1 IN POSITION 3 SUBSTITUTED-5-BETA-AMIDOMETHYL-OXAZOLIDIN-2-ONES THE UPJOHN COMPANY (US) 1990-03-22 WO disclosed
EP-0359418-A1 5'-Indolinyl-5beta-amidomethyloxazolidin-2-ones, 3-(fused-ring substituted)phenyl-5beta-amidomethyloxazolidin-2-ones and 3-(nitrogen substituted)phenyl-5beta-amidomethyloxazolidin-2-ones THE UPJOHN COMPANY (US) 1990-03-21 EP disclosed
EP-0311090-A1 Aminomethyl oxooxazolidinyl cycloalkylbenzene derivatives useful as antibacterial agents THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1989-04-12 EP disclosed
EP-0311090-A1 Aminomethyl oxooxazolidinyl cycloalkylbenzene derivatives useful as antibacterial agents THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1989-04-12 EP disclosed
US-4801600-A Aminomethyl oxooxazolidinyl cycloalkylbenzene derivatives useful as antibacterial agents E. I. DU PONT DE NEMOURS AND COMPANY (US) 1989-01-31 US disclosed
US-4801600-A Aminomethyl oxooxazolidinyl cycloalkylbenzene derivatives useful as antibacterial agents E. I. DU PONT DE NEMOURS AND COMPANY (US) 1989-01-31 US disclosed