SCHEMBL9450262

SCHEMBL9450262

C=C1c2cc(C(=O)OCC)ccc2CCC1c1ncc[nH]1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRA1A P35348 8/20 0.40
ALDH1A1 P00352 2/20 0.39
MAPK1 P28482 1/20 0.39
DRD3 P35462 2/20 0.38
DRD2 P14416 1/20 0.38
MAPT P10636 2/20 0.38
KDM4E B2RXH2 1/20 0.38
NPC1 O15118 1/20 0.38
LMNA P02545 1/20 0.38
HSD17B10 Q99714 1/20 0.38
IMPDH2 P12268 1/20 0.38
ADRA2A P08913 3/20 0.38
BRD4 O60885 1/20 0.37
GAA P10253 1/20 0.37
HTT P42858 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
CYP3A4 P08684 1/20 0.36
ADORA2A P29274 1/20 0.36
ADORA2B P29275 1/20 0.36
ALOX15 P16050 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9450073 0.73 ALDH1A1 (0.41) ALDH1A1MAPK1DRD3DRD2MAPT
SCHEMBL10532562 0.71 DRD3 (0.45) ALDH1A1MAPK1DRD3DRD2MAPT
SCHEMBL10531165 0.71 HTR2B (0.41) ALDH1A1MAPK1DRD3DRD2MAPT
Hydrochloric Acid SCHEMBL10531205 0.70 DRD3 (0.44) ALDH1A1MAPK1DRD3DRD2MAPT
SCHEMBL9450209 0.69 HTR2B (0.41) ALDH1A1KDM4ELMNA
SCHEMBL10528728 0.68 HTR2B (0.41) ALDH1A1MAPK1DRD3DRD2MAPT
SCHEMBL30782284 0.67 MAPK1 (0.57) ALDH1A1MAPK1MAPTKDM4ENPC1
SCHEMBL27145774 0.67 MAPK1 (0.57) ALDH1A1MAPK1MAPTKDM4ENPC1
SCHEMBL9812347 0.67 KDM4E (0.41) ALDH1A1MAPK1MAPTKDM4ENPC1
SCHEMBL30583381 0.67 BRD4 (0.55) ALDH1A1MAPK1MAPTKDM4ENPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5204364-A Selective inhibition of thromboxane A2; anticholesterol agents treating nephrosis, hyperlipidemia FARMITALIA CARLO ERBA, S.R.L. (IT) 1993-04-20 US disclosed
EP-0363789-B1 N-IMIDAZOLYL-AND N-IMIDAZOLYL-METHYL DERIVATIVES OR SUBSTITUTED BICYCLIC COMPOUNDS FARMITALIA CARLO ERBA S.r.l. (IT) 1992-05-06 EP disclosed
EP-0363789-A1 N-imidazolyl-and N-imidazolyl-methyl derivatives or substituted bicyclic compounds FARMITALIA CARLO ERBA S.r.l. (IT) 1990-04-18 EP disclosed