SCHEMBL9459052

SCHEMBL9459052

COC(=O)c1cc2c(s1)SCC2

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 8/20 0.49
HPGD P15428 7/20 0.49
KDM4E B2RXH2 6/20 0.49
MAPK1 P28482 5/20 0.49
L3MBTL1 Q9Y468 4/20 0.49
RAB9A P51151 2/20 0.49
NPC1 O15118 1/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
GAA P10253 3/20 0.46
ATM Q13315 3/20 0.46
GLA P06280 2/20 0.46
TDP1 Q9NUW8 2/20 0.46
MAPT P10636 2/20 0.46
TSHR P16473 3/20 0.42
CASP1 P29466 1/20 0.42
CASP7 P55210 1/20 0.42
HSD17B10 Q99714 1/20 0.42
CSNK2A2 P19784 1/20 0.38
KDR P35968 1/20 0.38
CSNK2B P67870 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9459054 0.82 ALDH1A1 (0.50) ALDH1A1HPGDKDM4EGLAMAPT
SCHEMBL6994905 0.73 KDM4E (0.39) ALDH1A1HPGDKDM4EMAPK1L3MBTL1
SCHEMBL15407033 0.71 DAO (0.69) ALDH1A1HPGDKDM4EMAPK1L3MBTL1
SCHEMBL13550064 0.71 KDM4E (0.66) ALDH1A1HPGDKDM4EMAPK1L3MBTL1
SCHEMBL7218427 0.71 ALDH1A1 (0.69) ALDH1A1HPGDKDM4EMAPK1L3MBTL1
SCHEMBL13550058 0.70 KDM4E (0.52) ALDH1A1HPGDKDM4EMAPK1L3MBTL1
SCHEMBL28870911 0.70 ALDH1A1 (0.67) ALDH1A1HPGDKDM4EMAPK1L3MBTL1
SCHEMBL12883525 0.70 ALDH1A1 (0.67) ALDH1A1HPGDKDM4EMAPK1L3MBTL1
SCHEMBL6995377 0.69 MAPT (0.41) ALDH1A1HPGDKDM4EMAPK1L3MBTL1
SCHEMBL13550073 0.69 KDM4E (0.48) ALDH1A1HPGDKDM4EMAPK1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5216020-A Antiglaucoma and occular hyptotensive agents MERCK & CO., INC. (US) 1993-06-01 US disclosed
EP-0480692-A2 Substituted 4,5-dihydrothieno[2,3-b]thiophene-2-sulfonamides MERCK & CO. INC. (US) 1992-04-15 EP disclosed