SCHEMBL945976

SCHEMBL945976

CC1=NC(c2cccc(-c3cccc(F)c3F)c2)(c2cnn(C)c2C)N=C1N

nearest known ligand 0.46

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 20/20 0.46
APP P05067 3/20 0.45
BACE2 Q9Y5Z0 2/20 0.44
CTSD P07339 1/20 0.44
KCNH2 Q12809 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL945867 0.83 BACE1 (0.43) BACE1APPBACE2CTSD
SCHEMBL946334 0.81 BACE1 (0.52) BACE1BACE2KCNH2
SCHEMBL945531 0.81 BACE1 (0.51) BACE1APPBACE2KCNH2
SCHEMBL943868 0.80 BACE1 (0.64) BACE1BACE2KCNH2
SCHEMBL945166 0.79 BACE1 (0.45) BACE1APPBACE2KCNH2
SCHEMBL944883 0.78 BACE1 (0.54) BACE1APPBACE2KCNH2
SCHEMBL932295 0.63 BACE1 (1.00) BACE1BACE2KCNH2
SCHEMBL948729 0.63 BACE1 (0.42) BACE1BACE2CTSDKCNH2
SCHEMBL932452 0.62 BACE1 (1.00) BACE1BACE2KCNH2
SCHEMBL9948389 0.62 BACE1 (1.00) BACE1APP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011002407-A1 NOVEL COMPOUNDS FOR TREATMENT OF NEURODEGENERATION ASSOCIATED WITH DISEASES, SUCH AS ALZHEIMER'S DISEASE OR DEMENTIA ASTRAZENECA AB (SE) 2011-01-06 WO disclosed
WO-2011002407-A1 NOVEL COMPOUNDS FOR TREATMENT OF NEURODEGENERATION ASSOCIATED WITH DISEASES, SUCH AS ALZHEIMER'S DISEASE OR DEMENTIA ASTRAZENECA AB (SE) 2011-01-06 WO disclosed