SCHEMBL945867

SCHEMBL945867

CC1=NC(c2cccc(-c3cccc(F)c3F)c2)(c2cnn(C)c2C)N=C1

nearest known ligand 0.43

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 18/20 0.43
BACE2 Q9Y5Z0 13/20 0.43
CTSD P07339 12/20 0.43
APP P05067 1/20 0.33
PGR P06401 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL945976 0.83 BACE1 (0.46) BACE1BACE2CTSDAPP
SCHEMBL948729 0.80 BACE1 (0.42) BACE1BACE2CTSD
SCHEMBL4527011 0.63 RPS6KA3 (0.45) BACE1APPPGR
SCHEMBL945531 0.62 BACE1 (0.51) BACE1BACE2APP
SCHEMBL945166 0.59 BACE1 (0.45) BACE1BACE2APP
SCHEMBL15344206 0.59 RAB9A (0.51)
SCHEMBL21324356 0.58 CHRM1 (0.48)
SCHEMBL3048969 0.57 TAAR1 (0.45) PGR
SCHEMBL2171711 0.56 CYP3A4 (0.46) BACE1APPPGR
SCHEMBL10091244 0.56 PGR (0.44) BACE1APPPGR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011002407-A1 NOVEL COMPOUNDS FOR TREATMENT OF NEURODEGENERATION ASSOCIATED WITH DISEASES, SUCH AS ALZHEIMER'S DISEASE OR DEMENTIA ASTRAZENECA AB (SE) 2011-01-06 WO claimed
WO-2011002407-A1 NOVEL COMPOUNDS FOR TREATMENT OF NEURODEGENERATION ASSOCIATED WITH DISEASES, SUCH AS ALZHEIMER'S DISEASE OR DEMENTIA ASTRAZENECA AB (SE) 2011-01-06 WO disclosed