SCHEMBL9466987

SCHEMBL9466987

C1=C(c2cccs2)CCN(CCCc2cnc3ccccc3c2)C1

nearest known ligand 0.61

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 7/20 0.61
PARP1 P09874 5/20 0.41
PPARG P37231 1/20 0.40
PPARA Q07869 1/20 0.40
TMEM97 Q5BJF2 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9467746 0.96 SIGMAR1 (0.65) SIGMAR1PARP1PPARGPPARA
SCHEMBL9467110 0.85 SIGMAR1 (0.58) SIGMAR1PARP1
Hydrochloric Acid SCHEMBL9719834 0.84 SIGMAR1 (0.57) SIGMAR1PARP1TMEM97
SCHEMBL8906589 0.84 SIGMAR1 (0.49) SIGMAR1
SCHEMBL9466847 0.82 SIGMAR1 (0.63) SIGMAR1PARP1
SCHEMBL9466984 0.81 SIGMAR1 (0.61) SIGMAR1PARP1
Hydrochloric Acid SCHEMBL9467616 0.81 SIGMAR1 (0.60) SIGMAR1PARP1
SCHEMBL10532112 0.80 SIGMAR1 (0.64) SIGMAR1PARP1
SCHEMBL9467634 0.79 SIGMAR1 (0.69) SIGMAR1PPARGPPARATMEM97
SCHEMBL9466973 0.76 SIGMAR1 (1.00) SIGMAR1PARP1PPARGPPARATMEM97

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5118691-A Substituted tetrahydropyridines as central nervous system agents WARNER-LAMBERT CO. (US) 1992-06-02 US claimed
US-5187280-A Dopaminergic, antipsychotic and antihypertensive agents WARNER-LAMBERT COMPANY (US) 1993-02-16 US disclosed
US-5118691-A Substituted tetrahydropyridines as central nervous system agents WARNER-LAMBERT CO. (US) 1992-06-02 US disclosed
US-5045550-A Antipsychotic, hypotensive agents, dopaminergic WARNER-LAMBERT CO. (US) 1991-09-03 US disclosed