SCHEMBL9467948

SCHEMBL9467948

COC(=O)C1=C(C)NC(C)=C(C#N)C1c1cccc2ncc(-c3ccccc3)cc12

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR3C2 P08235 5/20 0.62
CACNA1C Q13936 4/20 0.50
KDM4E B2RXH2 4/20 0.44
HSD17B10 Q99714 2/20 0.42
AXL P30530 2/20 0.42
ALDH1A1 P00352 2/20 0.42
MAPT P10636 2/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
CYP1A2 P05177 2/20 0.42
CYP3A4 P08684 2/20 0.42
CYP2C9 P11712 2/20 0.42
CYP2C19 P33261 2/20 0.42
MET P08581 1/20 0.42
ABCC4 O15439 1/20 0.42
PLIN1 O60240 1/20 0.42
CACNA1F O60840 1/20 0.42
GMNN O75496 1/20 0.42
KCNK2 O95069 1/20 0.42
ABCB11 O95342 1/20 0.42
GSR P00390 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9643618 0.91 NR3C2 (0.65) NR3C2CACNA1CCYP1A2CYP3A4CYP2C9
SCHEMBL9580964 0.90 CYP2C9 (0.51) NR3C2CACNA1CKDM4EHSD17B10AXL
SCHEMBL9644465 0.90 NR3C2 (0.77) NR3C2CACNA1CKDM4EMAPTCYP1A2
SCHEMBL9580965 0.88 CYP2C9 (0.48) NR3C2CACNA1CKDM4EHSD17B10AXL
SCHEMBL9463384 0.86 NR3C2 (0.54) NR3C2CACNA1CKDM4EHSD17B10AXL
SCHEMBL9463356 0.85 NR3C2 (0.47) NR3C2CACNA1CKDM4EHSD17B10ALDH1A1
SCHEMBL9140284 0.85 NR3C2 (0.44) NR3C2CACNA1CKDM4EHSD17B10AXL
SCHEMBL8923705 0.85 NR3C2 (0.52) NR3C2CACNA1CKDM4EALDH1A1MAPT
SCHEMBL7162892 0.85 NR3C2 (0.52) NR3C2CACNA1CKDM4EALDH1A1MAPT
SCHEMBL9468051 0.84 MAPT (0.56) NR3C2CACNA1CKDM4EHSD17B10AXL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5204472-A For preparing inotropic agents; substituted dihydropyridines BAYER AKTIENGESELLSCHAFT (DE) 1993-04-20 US disclosed
US-5100900-A Inotropic agents BAYER AKTIENGESELLSCHAFT (DE) 1992-03-31 US disclosed