SCHEMBL8923705

SCHEMBL8923705

CC1=C(C#N)C(c2cccc3ncc(-c4ccccc4)cc23)C(C(=O)O)=C(N)N1

nearest known ligand 0.52

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
NR3C2 P08235 5/20 0.52
MET P08581 2/20 0.41
CACNA1C Q13936 3/20 0.41
KDM4E B2RXH2 4/20 0.39
ALDH1A1 P00352 4/20 0.37
MAPT P10636 3/20 0.37
HTT P42858 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
THRB P10828 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7162892 1.00 NR3C2 (0.52) NR3C2METCACNA1CKDM4EALDH1A1
SCHEMBL27438736 0.90 CACNA1C (0.44) NR3C2METCACNA1CKDM4EALDH1A1
SCHEMBL6931471 0.89 NR3C2 (0.67) NR3C2METCACNA1CKDM4EALDH1A1
SCHEMBL7877495 0.89 NR3C2 (0.67) NR3C2METCACNA1CKDM4EALDH1A1
SCHEMBL9123412 0.87 NR3C2 (0.54) NR3C2CACNA1C
SCHEMBL9467948 0.85 NR3C2 (0.62) NR3C2METCACNA1CKDM4EALDH1A1
SCHEMBL9643618 0.83 NR3C2 (0.65) NR3C2CACNA1C
SCHEMBL7275395 0.83 NR3C2 (0.55) NR3C2METCACNA1CKDM4EALDH1A1
SCHEMBL9644465 0.83 NR3C2 (0.77) NR3C2METCACNA1CKDM4EMAPT
SCHEMBL9463271 0.81 NR3C2 (0.44) NR3C2METALDH1A1HTTNPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5653998-A Injectable liposomal pharmaceutical preparations BAYER AKTIENGESELLSCHAFT (DE) 1997-08-05 US disclosed
CN-1100418-A 2-amino-5-cyano-4-quinolyldihydropyridine esters, processes for their preparation and their use in medicaments BAYER AG (DE) 1995-03-22 CN disclosed