SCHEMBL9468337

SCHEMBL9468337

O=C(O)C=C(C(=O)O)c1ccc(Br)cc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.55
AKR1C3 P42330 2/20 0.49
CES2 O00748 1/20 0.48
CES1 P23141 1/20 0.48
CA1 P00915 2/20 0.45
CA2 P00918 2/20 0.45
PDPK1 O15530 1/20 0.44
ALDH1A1 P00352 1/20 0.43
MAPT P10636 1/20 0.43
GSK3B P49841 2/20 0.42
CYP1B1 Q16678 1/20 0.42
HAO1 Q9UJM8 1/20 0.42
OGG1 O15527 1/20 0.41
AKR1C1 Q04828 1/20 0.39
LMNA P02545 1/20 0.39
HDAC3 O15379 1/20 0.39
HDAC4 P56524 1/20 0.39
HDAC1 Q13547 1/20 0.39
HDAC7 Q8WUI4 1/20 0.39
HDAC2 Q92769 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9468335 1.00 CYP1A2 (0.55) CYP1A2AKR1C3CES2CES1CA1
SCHEMBL8743703 0.81 CPT1B (0.52) CYP1A2CES2CA1CA2ALDH1A1
SCHEMBL4771867 0.81 CYP1A2 (0.52) CYP1A2AKR1C3CES2CES1CA1
SCHEMBL4771865 0.81 CYP1A2 (0.52) CYP1A2AKR1C3CES2CES1CA1
SCHEMBL20366121 0.81 CPT1B (0.52) CYP1A2CES2CA1CA2ALDH1A1
SCHEMBL165294 0.80 AKR1C1 (0.59) AKR1C3CES2CES1CA1CA2
SCHEMBL164580 0.80 AKR1C1 (0.59) AKR1C3CES2CES1CA1CA2
SCHEMBL164579 0.80 AKR1C1 (0.59) AKR1C3CES2CES1CA1CA2
SCHEMBL9467960 0.79 ALDH1A1 (0.52) AKR1C3CES2CES1ALDH1A1MAPT
SCHEMBL9439222 0.79 ALDH1A1 (0.54) AKR1C3CES2CES1CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5206392-A Reacting arylacetonitriles with glyoxylic acid in presence of base, hydrolyzing, cyclizing AMERICAN CYANAMID COMPANY (US) 1993-04-27 US disclosed