SCHEMBL9469068

SCHEMBL9469068

Nc1ccncc1-c1cc2ccccc2[nH]1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 1/20 0.56
SLC22A12 Q96S37 1/20 0.52
GSK3B P49841 1/20 0.50
KDR P35968 4/20 0.49
CHEK1 O14757 1/20 0.49
RAB9A P51151 3/20 0.46
NPC1 O15118 2/20 0.46
KDM4E B2RXH2 3/20 0.45
MEN1 O00255 3/20 0.45
ALDH1A1 P00352 3/20 0.45
MAPT P10636 3/20 0.45
HPGD P15428 3/20 0.45
KMT2A Q03164 3/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
NPSR1 Q6W5P4 1/20 0.45
AOC3 Q16853 2/20 0.44
IDO1 P14902 1/20 0.44
TBK1 Q9UHD2 1/20 0.44
USP2 O75604 1/20 0.43
LMNA P02545 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1999798 0.81 KDM4E (0.57) CYP19A1SLC22A12GSK3BKDRCHEK1
SCHEMBL29361867 0.80 KDR (0.58) CYP19A1GSK3BKDRCHEK1RAB9A
SCHEMBL221259 0.80 KDR (0.58) CYP19A1GSK3BKDRCHEK1RAB9A
SCHEMBL1999569 0.78 CYP19A1 (0.56) CYP19A1SLC22A12GSK3BKDRCHEK1
SCHEMBL5207806 0.75 KDR (0.74) CYP19A1SLC22A12KDRCHEK1KDM4E
SCHEMBL4779547 0.75 KDR (0.74) CYP19A1SLC22A12KDRCHEK1KDM4E
SCHEMBL21727914 0.75 SLC22A12 (0.74) CYP19A1SLC22A12GSK3BKDRCHEK1
SCHEMBL26053442 0.74 KDR (0.51) CYP19A1SLC22A12GSK3BKDRCHEK1
SCHEMBL25166926 0.74 CYP19A1 (0.77) CYP19A1SLC22A12KDRCHEK1RAB9A
SCHEMBL7062756 0.74 SLC22A12 (0.57) CYP19A1SLC22A12KDRCHEK1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5214059-A Dermatitis, psoriasis HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1993-05-25 US claimed
US-5214059-A Dermatitis, psoriasis HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1993-05-25 US disclosed
US-5166170-A 2-(AMINOARYL) INDOLES AND INDOLINES AS TOPICAL ANTIINFLAMMATORY AGENTS FOR THE TREATMENT OF SKIN DISORDERS HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1992-11-24 US disclosed
EP-0406734-A2 2-(Aminoaryl)indoles and indolines, a process for their preparation and their use as medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1991-01-09 EP disclosed