SCHEMBL221259

SCHEMBL221259

Nc1ccccc1-c1cc2ccccc2[nH]1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 2/20 0.58
CHEK1 O14757 1/20 0.58
RAB9A P51151 5/20 0.57
KDM4E B2RXH2 5/20 0.57
MAPT P10636 5/20 0.57
ALDH1A1 P00352 5/20 0.57
HPGD P15428 4/20 0.57
MEN1 O00255 3/20 0.57
KMT2A Q03164 3/20 0.57
SMN1; SMN2 Q16637 2/20 0.57
NPSR1 Q6W5P4 2/20 0.57
NPC1 O15118 4/20 0.55
AOC3 Q16853 2/20 0.53
GAA P10253 2/20 0.50
HSD17B10 Q99714 2/20 0.50
USP2 O75604 1/20 0.50
LMNA P02545 1/20 0.50
POLB P06746 1/20 0.50
ALOX15 P16050 1/20 0.50
TDP1 Q9NUW8 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29361867 1.00 KDR (0.58) KDRCHEK1RAB9AKDM4EMAPT
SCHEMBL3138805 0.87 KDR (0.53) KDRCHEK1RAB9AKDM4EMAPT
SCHEMBL5051826 0.86 KDR (0.68) KDRCHEK1RAB9AKDM4EMAPT
SCHEMBL2563486 0.84 KDR (0.53) KDRCHEK1RAB9AKDM4EMAPT
SCHEMBL29733654 0.84 KDR (0.53) KDRCHEK1RAB9AKDM4EMAPT
SCHEMBL29419326 0.84 KDR (0.53) KDRCHEK1RAB9AKDM4EMAPT
Methane SCHEMBL28704887 0.84 KDR (0.66) KDRCHEK1RAB9AKDM4EMAPT
Benzene SCHEMBL27629233 0.84 RAB9A (0.69) KDRCHEK1RAB9AKDM4EMAPT
SCHEMBL8965829 0.82 RAB9A (0.58) KDRCHEK1RAB9AKDM4EMAPT
Hydrochloric Acid SCHEMBL3675763 0.82 KDR (0.51) KDRCHEK1RAB9AKDM4EMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 285 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114621220-B Indolo [3,2-c ] quinoline compound and synthesis method thereof 无锡学院 2023-07-04 CN claimed
CN-114621220-A Indolo [3,2-c ] quinoline compound and synthetic method thereof 无锡学院 2022-06-14 CN claimed
CN-108424416-B Method for synthesizing indole [1,2-c ] quinazoline compound 河南师范大学 2021-04-16 CN claimed
US-6656237-B1 Fused polycyclic aromatic compound with exocyclic nitrogen group attached directly to a ring carbon; 1-amino naphthalene, 1,8-diaminonaphthalene, 5-aminoindole, 2-(2-aminophenyl) indole, 8-aminoquinoline EXXONMOBIL RESEARCH AND ENGINEERING COMPANY 2003-12-02 US claimed
EP-1137746-A1 FUEL COMPOSITION WITH IMPROVED LUBRICITY PERFORMANCE ExxonMobil Research and Engineering Company (US) 2001-10-04 EP claimed
WO-2001021739-A1 FUEL COMPOSITION WITH IMPROVED LUBRICITY PERFORMANCE EXXONMOBIL RESEARCH AND ENGINEERING COMPANY (US) 2001-03-29 WO claimed
US-20240124404-A1 COMPOSITION FOR TREATING DISEASES RELATED TO ADVANCED GLYCATION END PRODUCTS COMPRISING INDOLE DERIVATIVE METACEN THERAPEUTICS (KR) 2024-04-18 US disclosed
EP-4353227-A1 COMPOSITION INCLUDING INDOLE DERIVATIVE FOR PREVENTION OF ADVANCED GLYCATION END PRODUCT-RELATED DISEASE Metacen Therapeutics (KR) 2024-04-17 EP disclosed
CN-114621220-B Indolo [3,2-c ] quinoline compound and synthesis method thereof 无锡学院 2023-07-04 CN disclosed
CN-114621220-B Indolo [3,2-c ] quinoline compound and synthesis method thereof 无锡学院 2023-07-04 CN disclosed
US-11678576-B2 Heterocyclic compound and organic light emitting element comprising same LT MATERIALS CO., LTD. (KR) 2023-06-13 US disclosed
CN-111253583-B Dilatant hybrid dynamic polymer and dilatant realization method thereof 厦门天策材料科技有限公司 2023-05-16 CN disclosed
CN-114621220-A Indolo [3,2-c ] quinoline compound and synthetic method thereof 无锡学院 2022-06-14 CN disclosed
US-5214059-A Dermatitis, psoriasis HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1993-05-25 US disclosed
US-5166170-A 2-(AMINOARYL) INDOLES AND INDOLINES AS TOPICAL ANTIINFLAMMATORY AGENTS FOR THE TREATMENT OF SKIN DISORDERS HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1992-11-24 US disclosed
US-5045539-A 1H-indolo[3,2-c]quinoline-derivatives, compositions containing same, useful for treating pain, psychosis or convulsions HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1991-09-03 US disclosed
US-5006531-A 5,6-dihydro(1H-indolo(3,2-C)quinoline-6,4'-piperidines) and related compounds which are useful for treating pain, psychosis or convulsions HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1991-04-09 US disclosed
EP-0407898-A1 5,6-dihydro(1H-indolo(3,2-c)quinoline-6,4-piperidines)and related compounds, a process for their preparation and their use as medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1991-01-16 EP disclosed
EP-0406734-A2 2-(Aminoaryl)indoles and indolines, a process for their preparation and their use as medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1991-01-09 EP disclosed
US-4057530-A STABILIZERS FOR VINYL CHLORIDE POLYMERS LABAZ (FR) 1977-11-08 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240124404-A1 COMPOSITION FOR TREATING DISEASES RELATED TO ADVANCED GLYCATION END PRODUCTS COMPRISING INDOLE DERIVATIVE AGER, IDO1, IAPP KDR 4006/4885CHEK1 3503/4885RAB9A 3408/4885
US-11678576-B2 Heterocyclic compound and organic light emitting element comprising same CRY1, CRY2, CYP1A1 KDR 2641/4885CHEK1 1843/4885RAB9A 2438/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.