SCHEMBL9475159

SCHEMBL9475159

CC(Br)c1ccccc1.O=S(=O)(Cl)Cl

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES2 O00748 1/20 0.41
CES1 P23141 1/20 0.41
ALDH1A1 P00352 3/20 0.41
TDP1 Q9NUW8 2/20 0.41
HSD17B10 Q99714 1/20 0.41
KDM4E B2RXH2 1/20 0.40
GMNN O75496 1/20 0.40
LMNA P02545 1/20 0.40
POLB P06746 1/20 0.40
MAPT P10636 1/20 0.40
HPGD P15428 1/20 0.40
PMP22 Q01453 1/20 0.40
KMT2A Q03164 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
TAAR1 Q96RJ0 3/20 0.39
TSHR P16473 1/20 0.39
SRC P12931 1/20 0.38
TRPA1 O75762 1/20 0.37
ADRA2A P08913 1/20 0.35
ADRA2C P18825 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4710 0.85
SCHEMBL1551 0.85
Benzene SCHEMBL22288204 0.85 TAAR1 (0.48) CES2CES1ALDH1A1KDM4ELMNA
SCHEMBL14127281 0.85
SCHEMBL3728 0.85
Iodide SCHEMBL27892619 0.83 TAAR1 (0.46) CES2CES1ALDH1A1KDM4ELMNA
SCHEMBL11031524 0.83 TAAR1 (0.46) CES2CES1ALDH1A1KDM4ELMNA
Bromide SCHEMBL28665198 0.83 TAAR1 (0.46) CES2CES1ALDH1A1KDM4ELMNA
SCHEMBL3226267 0.83 TAAR1 (0.46) CES2CES1ALDH1A1KDM4ELMNA
Isopropylbenzene SCHEMBL1416132 0.81 ALDH1A1 (0.44) ALDH1A1TDP1HSD17B10KDM4EGMNN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 19 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104903291-A Benzyl sulfonamide derivatives as RORc modulators HOFFMANN LA ROCHE 2015-09-09 CN disclosed
CN-102264704-B Isoquinoline derivative TAISHO PHARMACEUTICAL CO LTD 2014-06-04 CN disclosed
CN-103827117-A Tetrahydrotriazolopyrimidine derivatives as human neutrophil elastase inhibitors CHIESI FARMA SPA 2014-05-28 CN disclosed
CN-101268070-B Novel sulphonylpyrroles as inhibitors of HDAC novel sulphonylpyrroles NYCOMED GMBH 2012-09-05 CN disclosed
CN-102329267-A 6-substituted 2,3,4, 5-tetrahydro-1H-benzo [d] aza as 5-HT2Creceptor agonists LILLY CO ELI 2012-01-25 CN disclosed
CN-102311387-A 6-substituted 2,3,4, 5-tetrahydro-1H-benzo [d] aza as 5-HT2Creceptor agonists LILLY CO ELI 2012-01-11 CN disclosed
CN-102282143-A Heterocyclically substituted aryl compounds and application thereof 2011-12-14 CN disclosed
CN-102264704-A Isoquinoline derivative 2011-11-30 CN disclosed
CN-102056905-A Novel uracil compound having human deoxyuridine triphosphatase inhibitory activity or salt thereof TAIHO PHARMACEUTICAL CO LTD 2011-05-11 CN disclosed
CN-1918155-B Compounds and compositions as LXR modulators IRM LLC 2010-05-26 CN disclosed
CN-101287706-A Sulphonylpyrrole hydrochloride salts as histone deacetylases inhibitors NYCOMED GMBH (DE) 2008-10-15 CN disclosed
CN-101268070-A Novel sulphonylpyrroles as inhibitors of HDAC novel sulphonylpyrroles NYCOMED GMBH (DE) 2008-09-17 CN disclosed
CN-1934088-A As 5-HT2c6-substituted 2,3,4, 5-tetrahydro-1H-benzo [ d ] receptor agonists]Aza * LILLY CO ELI (US) 2007-03-21 CN disclosed
CN-1918155-A Compounds and compositions as lxr modulators IRM LLC (BM) 2007-02-21 CN disclosed
CN-1290254-A Sulfonamide derivatives process for producing the same and utilization thereof TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2001-04-04 CN disclosed
CN-1080923-A Benzo pyridone and pyridopyridine ketone that Sulphonylbenzyl replaces BAYER AG (DE) 1994-01-19 CN disclosed
CN-1077710-A The imidazoles that Sulphonylbenzyl replaces BAYED AG (DE) 1993-10-27 CN disclosed
CN-1077195-A The imidazopyridine that has replaced Sulphonylbenzyl BAYER AG (DE) 1993-10-13 CN disclosed
US-5203982-A Electrodialysis IONICS, INCORPORATED (US) 1993-04-20 US disclosed