SCHEMBL9476232

SCHEMBL9476232

CCCCCCc1cnc(C(=O)O)nc1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RARB P10826 6/20 0.63
ALDH1A1 P00352 3/20 0.54
MAPT P10636 3/20 0.54
NFKB1 P19838 2/20 0.54
MEN1 O00255 2/20 0.54
KMT2A Q03164 2/20 0.54
KDM4E B2RXH2 1/20 0.54
LMNA P02545 1/20 0.54
CYP1A2 P05177 1/20 0.54
CYP3A4 P08684 1/20 0.54
PKM P14618 1/20 0.54
ALOX15 P16050 1/20 0.54
TSHR P16473 1/20 0.54
THPO P40225 1/20 0.54
BLM P54132 1/20 0.54
PMP22 Q01453 1/20 0.54
HIF1A Q16665 1/20 0.54
TDP1 Q9NUW8 1/20 0.54
L3MBTL1 Q9Y468 1/20 0.54
NPC1 O15118 2/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9476450 1.00 RARB (0.63) RARBALDH1A1MAPTNFKB1MEN1
SCHEMBL9476466 1.00 RARB (0.63) RARBALDH1A1MAPTNFKB1MEN1
SCHEMBL10335865 0.98 RARB (0.60) RARBALDH1A1MAPTNFKB1MEN1
SCHEMBL9233439 0.93 ALDH1A1 (0.62) RARBALDH1A1MAPTNFKB1MEN1
SCHEMBL9478086 0.85 SMN1; SMN2 (0.50) RARBALDH1A1MAPTNFKB1MEN1
SCHEMBL14028771 0.84 RARB (0.54) RARBALDH1A1MAPTNFKB1MEN1
SCHEMBL9453893 0.84 RARB (0.54) RARBALDH1A1MAPTNFKB1MEN1
SCHEMBL10986992 0.78 ALDH1A1 (0.88) RARBALDH1A1MAPTNFKB1MEN1
SCHEMBL10662786 0.78 ALDH1A1 (0.88) RARBALDH1A1MAPTNFKB1MEN1
SCHEMBL10359434 0.78 RARB (0.55) RARBALDH1A1MAPTNFKB1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9714240-B2 Vinyl autotaxin inhibitor compounds PHARMAKEA, INC. (US) 2017-07-25 US disclosed
US-5182047-A FLUORINATED BIPHENYLDIOLE DERIVATIVES MERCK PATENT GESELLSCHAFT MIT BESCHRAENKTER HAFTUNG (DE) 1993-01-26 US disclosed
EP-0368975-A1 FLUORINATED BIPHENYLDIOLE DERIVATIVES. MERCK PATENT GMBH (DE) 1990-05-23 EP disclosed
WO-1989012039-A1 FLUORINATED BIPHENYLDIOLE DERIVATIVES MERCK Patent Gesellschaft mit beschränkter Haftung (DE) 1989-12-14 WO disclosed