SCHEMBL9476489

SCHEMBL9476489

COC(=O)C1(C)Cc2c([nH]c3ccccc23)CN1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.50
CYP1A2 P05177 2/20 0.50
CYP2D6 P10635 2/20 0.50
CYP2C9 P11712 2/20 0.50
CYP2C19 P33261 2/20 0.50
HSD17B10 Q99714 2/20 0.50
MAPT P10636 2/20 0.50
ALDH1A1 P00352 1/20 0.50
GAA P10253 1/20 0.50
HPGD P15428 1/20 0.50
ALOX15 P16050 1/20 0.50
CYP19A1 P11511 4/20 0.43
HTR5A P47898 1/20 0.41
NISCH Q9Y2I1 1/20 0.41
NR2E1 Q9Y466 1/20 0.41
MAPK1 P28482 1/20 0.41
IDO1 P14902 1/20 0.41
PTPN1 P18031 1/20 0.41
PDE5A O76074 2/20 0.41
LMNA P02545 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1520201 0.85 KDM4E (0.44) KDM4ECYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL31280140 0.77 KDM4E (0.50) KDM4ECYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL9845301 0.76 KDM4E (0.44) KDM4ECYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL999715 0.74 KDM4E (0.50) KDM4ECYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL5881088 0.72 TACR1 (0.66) KDM4ECYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL27927974 0.72 MEN1 (0.44) KDM4ECYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL997234 0.72 KDM4E (0.47) KDM4ECYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL997617 0.72 KDM4E (0.47) KDM4ECYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL6238822 0.70 KMT2A (0.51) KDM4ECYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL21043206 0.70 KDM4E (0.38) KDM4ECYP1A2CYP2D6CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5244905-A Gastric antisecretory, antipsychotic, appetite suppressants WARNER-LAMBERT COMPANY (US) 1993-09-14 US disclosed
WO-1992004348-A1 N-SUBSTITUTED CYCLOALKYL AND POLYCYCLOAKYL POLYHYDRO-Β-CARBOLINE-PHENYLALANINE-AND PHENETHYLAMINE DERIVATIVES WARNER-LAMBERT COMPANY (US) 1992-03-19 WO disclosed