SCHEMBL9477146

SCHEMBL9477146

CCCCOc1ccc(-c2ccc(OC(C)C(=O)O)cc2)cc1F

nearest known ligand 0.52

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.52
GAA P10253 1/20 0.52
CYP2C9 P11712 1/20 0.52
PKM P14618 1/20 0.52
CYP2C19 P33261 1/20 0.52
RARB P10826 2/20 0.51
RARA P10276 1/20 0.51
PPARD Q03181 3/20 0.45
PPARG P37231 2/20 0.45
PPARA Q07869 2/20 0.45
S1PR1 P21453 1/20 0.45
PTPN11 Q06124 2/20 0.44
FFAR1 O14842 2/20 0.44
NR1H4 Q96RI1 1/20 0.44
FFAR4 Q5NUL3 3/20 0.43
TDP1 Q9NUW8 1/20 0.43
MAP4K4 O95819 2/20 0.42
PTPN1 P18031 1/20 0.42
PTPN6 P29350 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9476529 0.98 CYP1A2 (0.50) CYP1A2GAACYP2C9PKMCYP2C19
SCHEMBL9475785 0.96 PTPN11 (0.50) CYP1A2GAACYP2C9PKMCYP2C19
SCHEMBL9477572 0.96 PTPN11 (0.50) CYP1A2GAACYP2C9PKMCYP2C19
SCHEMBL9476709 0.96 PTPN11 (0.50) CYP1A2GAACYP2C9PKMCYP2C19
SCHEMBL9475444 0.95 CYP1A2 (0.52) CYP1A2GAACYP2C9PKMCYP2C19
SCHEMBL9475894 0.90 CYP1A2 (0.55) CYP1A2GAACYP2C9PKMCYP2C19
SCHEMBL9399442 0.81 S1PR1 (0.51) CYP1A2CYP2C9CYP2C19RARBRARA
SCHEMBL8881964 0.80 RARB (0.62) CYP1A2GAACYP2C9PKMCYP2C19
SCHEMBL9399572 0.80 S1PR1 (0.49) CYP1A2CYP2C9CYP2C19RARBRARA
SCHEMBL9478161 0.79 RARA (0.41) RARBRARAS1PR1PTPN11FFAR4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5182047-A FLUORINATED BIPHENYLDIOLE DERIVATIVES MERCK PATENT GESELLSCHAFT MIT BESCHRAENKTER HAFTUNG (DE) 1993-01-26 US disclosed