SCHEMBL9485441

SCHEMBL9485441

CC(C(=O)O)c1ccncc1.NC(=O)Cc1ccncc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 5/20 0.46
PTGS1 P23219 4/20 0.46
AKR1C3 P42330 3/20 0.46
LMNA P02545 2/20 0.46
CYP2C9 P11712 2/20 0.46
CXCR1 P25024 2/20 0.46
CXCR2 P25025 2/20 0.46
AKR1C2 P52895 2/20 0.46
ALB P02768 1/20 0.46
ESR1 P03372 1/20 0.46
ALOX5 P09917 1/20 0.46
RARB P10826 1/20 0.46
ADRB3 P13945 1/20 0.46
NFKB1 P19838 1/20 0.46
HTR2A P28223 1/20 0.46
NR1I3 Q14994 1/20 0.46
SLC22A6 Q4U2R8 1/20 0.46
CXCL8 P10145 1/20 0.46
TSHR P16473 1/20 0.46
BLM P54132 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14537418 0.83 AKR1C3 (0.56) PTGS2PTGS1AKR1C3LMNACYP2C9
SCHEMBL1690400 0.83 AKR1C3 (0.56) PTGS2PTGS1AKR1C3LMNACYP2C9
Hydrochloric Acid SCHEMBL8937692 0.81 AKR1C3 (0.54) PTGS2PTGS1AKR1C3LMNACYP2C9
SCHEMBL1178369 0.81 CA2 (0.58) CYP19A1RAB9ASMN1; SMN2CA2
Hydrochloric Acid SCHEMBL2673007 0.79 CA2 (0.56) CYP19A1RAB9ASMN1; SMN2CA2
SCHEMBL9484991 0.76 NAPRT (0.53) AKR1C3LMNACYP2C9AKR1C2ESR1
SCHEMBL5509666 0.74 CYP17A1 (0.61) TSHRCYP19A1RAB9ASMN1; SMN2CA2
SCHEMBL28156856 0.74 CA2 (0.50) CYP19A1RAB9ASMN1; SMN2CA2SLC22A12
SCHEMBL2371076 0.74 EPHX1 (0.53) PTGS2AKR1C3CYP2C9AKR1C2CYP19A1
SCHEMBL7767500 0.74 EPHX1 (0.53) PTGS2AKR1C3CYP2C9AKR1C2CYP19A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0525109-A4 STYRYL-SUBSTITUTED MONOCYCLIC AND BICYCLIC HETEROARYL COMPOUNDS WHICH INHIBIT EGF RECEPTOR TYROSINE KINASE 1993-06-30 EP disclosed
EP-0525109-A1 STYRYL-SUBSTITUTED MONOCYCLIC AND BICYCLIC HETEROARYL COMPOUNDS WHICH INHIBIT EGF RECEPTOR TYROSINE KINASE RHONE-POULENC RORER INTERNATIONAL (HOLDINGS) INC. (US) 1993-02-03 EP disclosed