SCHEMBL9488146

SCHEMBL9488146

CCc1ccc([N+](=O)[O-])c(Br)c1

nearest known ligand 0.49

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KAT2B Q92831 1/20 0.49
KMT2A Q03164 3/20 0.43
CYP19A1 P11511 5/20 0.43
LMNA P02545 4/20 0.43
MAPT P10636 3/20 0.43
HTT P42858 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
AAK1 Q2M2I8 1/20 0.42
CYP3A4 P08684 2/20 0.41
TSHR P16473 1/20 0.41
ALDH1A1 P00352 5/20 0.41
MEN1 O00255 2/20 0.41
GAA P10253 1/20 0.41
ALPG P10696 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
CYP2D6 P10635 1/20 0.39
CYP1A2 P05177 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28671318 0.86 CYP19A1 (0.43) KAT2BCYP19A1MAPTAAK1CYP3A4
SCHEMBL278730 0.85 ALDH1A1 (0.50) KAT2BKMT2ALMNAMAPTHTT
SCHEMBL3649190 0.83 CYP19A1 (0.46) CYP19A1MAPTAAK1CYP3A4TSHR
SCHEMBL10959235 0.82 TSHR (0.55) KAT2BKMT2ALMNAMAPTHTT
SCHEMBL27748882 0.81 CYP19A1 (0.43) KMT2ACYP19A1LMNAMAPTAAK1
SCHEMBL15248984 0.81 ALDH1A1 (0.47) CYP19A1MAPTAAK1CYP3A4TSHR
SCHEMBL13344089 0.81 KAT2B (0.48) KAT2BKMT2ALMNAMAPTHTT
SCHEMBL31449975 0.81 CYP19A1 (0.40) KMT2ACYP19A1LMNAMAPTSMN1; SMN2
SCHEMBL28676747 0.80 KCNH2 (0.48) LMNACYP3A4ALDH1A1
SCHEMBL4313888 0.80 CYP19A1 (0.42) CYP19A1AAK1CYP3A4TSHRALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011087738-A2 1,4-SUBSTITUTED PIPERAZINE DERIVATIVES AND METHODS OF USE THEREOF SCHERING CORPORATION (US) 2011-07-21 WO disclosed
EP-0325892-B1 PROCESS FOR THE PREPARATION OF HALOGENATED PRIMARY AMINES CIBA-GEIGY AG (CH) 1993-02-03 EP disclosed
EP-0473552-A1 Process for the preparation of halogenated aromatic primary amines CIBA-GEIGY AG (CH) 1992-03-04 EP disclosed
US-4960936-A Process for the preparation of halogenated aromatic primary amines CIBA-GEIGY CORPORATION (US) 1990-10-02 US disclosed
EP-0325892-A2 Process for the preparation of halogenated primary amines CIBA-GEIGY AG (CH) 1989-08-02 EP disclosed