SCHEMBL9493013

SCHEMBL9493013

CCOC(=O)CC(C)N1C(=O)c2cc(CCC(=O)NCCNC(=O)OC(C)(C)C)ccc2N(C)C(=O)C1c1ccccc1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDCD1 Q15116 1/20 0.37
CD274 Q9NZQ7 1/20 0.37
SCN9A Q15858 3/20 0.35
SIGMAR1 Q99720 2/20 0.34
CCKBR P32239 2/20 0.33
SLC6A9 P48067 1/20 0.33
ALDH1A1 P00352 2/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
LMNA P02545 1/20 0.33
HDAC3 O15379 2/20 0.33
HDAC1 Q13547 2/20 0.33
HDAC8 Q9BY41 2/20 0.33
HDAC6 Q9UBN7 2/20 0.33
HDAC4 P56524 1/20 0.33
HDAC7 Q8WUI4 1/20 0.33
HDAC2 Q92769 1/20 0.33
HDAC10 Q969S8 1/20 0.33
HDAC11 Q96DB2 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9493733 0.92 PDCD1 (0.36) PDCD1CD274SCN9ASIGMAR1CCKBR
SCHEMBL9492960 0.92 PDCD1 (0.38) PDCD1CD274SIGMAR1SLC6A9ALDH1A1
SCHEMBL9493816 0.91 PDCD1 (0.36) PDCD1CD274SIGMAR1ALDH1A1CYP3A4
SCHEMBL7326347 0.91 TPSAB1 (0.37) PDCD1CD274SCN9ASIGMAR1CCKBR
SCHEMBL7331594 0.89 NR1H2 (0.34) SCN9ASLC6A9MDM2
SCHEMBL9494267 0.85 PDCD1 (0.36) PDCD1CD274SCN9ASIGMAR1CYP3A4
SCHEMBL9264467 0.85 MDM2 (0.34) PDCD1CD274SCN9ACCKBRCCKAR
SCHEMBL7332035 0.84 SCN9A (0.39) SCN9ACCKBRCCKARMDM2
SCHEMBL9493769 0.84 PDCD1 (0.37) PDCD1CD274SIGMAR1CYP3A4CYP2C9
SCHEMBL7326646 0.83 TPSAB1 (0.36) PDCD1CD274SCN9ASIGMAR1TPSAB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5250679-A Nonpeptidyl platelet aggregation inhibitors having specificity for the GPIIb III.sub. receptor GENENTECH, INC. (US) 1993-10-05 US disclosed