SCHEMBL9494192

SCHEMBL9494192

Cc1cc(O)c2cc(C(F)(F)F)ccc2n1

nearest known ligand 0.50

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
GAK O14976 1/20 0.50
KDM4E B2RXH2 1/20 0.47
CCNE2 O96020 1/20 0.46
CCNA2 P20248 1/20 0.46
CCNE1 P24864 1/20 0.46
CDK2 P24941 1/20 0.46
CCNA1 P78396 1/20 0.46
DHODH Q02127 2/20 0.45
MCHR1 Q99705 1/20 0.44
RIPK2 O43353 1/20 0.42
KDR P35968 1/20 0.42
MAPK14 Q16539 1/20 0.42
SORT1 Q99523 1/20 0.42
CYP1A2 P05177 1/20 0.41
BACE1 P56817 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL899555 0.87 KDM4E (0.47) GAKKDM4ESORT1CYP1A2
SCHEMBL29588619 0.83 CYP1A2 (0.56) GAKKDM4ECCNE2CCNA2CCNE1
SCHEMBL19983427 0.83 CYP1A2 (0.56) GAKKDM4ECCNE2CCNA2CCNE1
SCHEMBL2712104 0.81 KDM4E (0.49) KDM4ECCNE2CCNA2CCNE1CDK2
SCHEMBL5101813 0.80 LMNA (0.62) GAKCCNE2CCNA2CCNE1CDK2
SCHEMBL12033714 0.80 KDM4E (0.47) GAKKDM4ECCNE2CCNA2CCNE1
SCHEMBL437638 0.80 MCHR1 (0.59) GAKMCHR1BACE1
SCHEMBL21173342 0.78 GAK (0.48) GAKKDM4ECCNE2CCNA2CCNE1
SCHEMBL3906125 0.77 GAA (0.47) KDM4EDHODHCYP1A2
SCHEMBL3760247 0.77 LMNA (0.61) KDM4ECYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0113432-B1 CHLOROMETHYL QUINOLINE DERIVATIVES, PROCESS FOR THEIR PREPARATION AND THEIR USE ALKALOIDA VEGYéSZETI GYáR (HU) 1993-03-17 EP disclosed
EP-0113432-A1 Chloromethyl quinoline derivatives, process for their preparation and their use ALKALOIDA VEGYéSZETI GYáR (HU) 1984-07-18 EP disclosed