SCHEMBL9495802

SCHEMBL9495802

CCc1ccc(C#Cc2ccc(C)cn2)cc1

nearest known ligand 0.53

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ACACB O00763 6/20 0.46
FFAR1 O14842 1/20 0.42
FFAR4 Q5NUL3 1/20 0.42
GRM5 P41594 3/20 0.41
CYP2A6 P11509 1/20 0.40
EGLN1 Q9GZT9 1/20 0.39
MCHR1 Q99705 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9855660 0.88 EGLN1 (0.48) ACACBFFAR1FFAR4GRM5CYP2A6
SCHEMBL9494958 0.88 ACACB (0.49) ACACBFFAR1FFAR4GRM5CYP2A6
SCHEMBL9500122 0.87 ACACB (0.44) ACACBFFAR1FFAR4GRM5MCHR1
SCHEMBL14129682 0.86 GRM5 (0.53) ACACBGRM5
SCHEMBL9498756 0.84 MCHR1 (0.44) ACACBFFAR1FFAR4MCHR1
SCHEMBL9499796 0.83 MCHR1 (0.44) ACACBFFAR1FFAR4MCHR1
SCHEMBL9496080 0.82 HSD17B10 (0.46) ACACBFFAR1FFAR4MCHR1
SCHEMBL9496532 0.82 HSD17B10 (0.46) ACACBFFAR1FFAR4MCHR1
SCHEMBL9495618 0.82 HSD17B10 (0.46) ACACBFFAR1FFAR4MCHR1
SCHEMBL9495556 0.82 ACACB (0.54) ACACBGRM5MCHR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0306505-B1 ACETYLENE DERIVATIVES AS COMPONENTS OF LIQUID CRYSTAL PHASES MERCK PATENT GmbH (DE) 1993-03-24 EP disclosed
EP-0306505-A1 ACETYLENE DERIVATIVES AS COMPONENTS OF LIQUID CRYSTAL PHASES. MERCK PATENT GMBH (DE) 1989-03-15 EP disclosed
WO-1988007523-A1 ACETYLENE DERIVATIVES AS COMPONENTS OF LIQUID CRYSTAL PHASES MERCK Patent Gesellschaft mit beschränkter Haftung (DE) 1988-10-06 WO disclosed