SCHEMBL9497535

SCHEMBL9497535

CC1CCC(C#Cc2ccc(-c3ccc(C#N)cc3)cc2)CC1

nearest known ligand 0.45

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 16/20 0.45
HRH2 P25021 4/20 0.45
HRH1 P35367 4/20 0.45
KIF11 P52732 1/20 0.41
MMP3 P08254 1/20 0.40
KCNH2 Q12809 2/20 0.40
FFAR1 O14842 1/20 0.39
HSD11B1 P28845 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9497527 1.00 HRH3 (0.45) HRH3HRH2HRH1KIF11MMP3
SCHEMBL9855720 0.90 FFAR1 (0.39) HRH3HRH2HRH1KCNH2FFAR1
SCHEMBL9498836 0.90 FFAR1 (0.39) HRH3HRH2HRH1KCNH2FFAR1
SCHEMBL9498830 0.90 FFAR1 (0.39) HRH3HRH2HRH1KCNH2FFAR1
SCHEMBL21258030 0.86 FFAR1 (0.47) HRH3MMP3FFAR1
SCHEMBL29306016 0.83 APP (0.42) HRH3FFAR1
SCHEMBL9495626 0.83 HRH3 (0.41) HRH3HRH2HRH1KIF11MMP3
SCHEMBL9495632 0.83 HRH3 (0.41) HRH3HRH2HRH1KIF11MMP3
SCHEMBL10513499 0.81 FFAR1 (0.36) HRH3HRH2HRH1FFAR1HSD11B1
SCHEMBL9495948 0.80 HRH3 (0.40) HRH3HRH2HRH1KIF11KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0306505-B1 ACETYLENE DERIVATIVES AS COMPONENTS OF LIQUID CRYSTAL PHASES MERCK PATENT GmbH (DE) 1993-03-24 EP disclosed
US-5068053-A Liquid crystals for optical apparatus MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1991-11-26 US disclosed
EP-0306505-A1 ACETYLENE DERIVATIVES AS COMPONENTS OF LIQUID CRYSTAL PHASES. MERCK PATENT GMBH (DE) 1989-03-15 EP disclosed
WO-1988007523-A1 ACETYLENE DERIVATIVES AS COMPONENTS OF LIQUID CRYSTAL PHASES MERCK Patent Gesellschaft mit beschränkter Haftung (DE) 1988-10-06 WO disclosed