SCHEMBL9499428

SCHEMBL9499428

CCc1ccc(C#Cc2ccc(Cl)cn2)cc1

nearest known ligand 0.51

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 6/20 0.48
ACACB O00763 5/20 0.42
CHRM1 P11229 2/20 0.41
HTR2A P28223 2/20 0.41
CYP2D6 P10635 1/20 0.41
FFAR1 O14842 1/20 0.41
FFAR4 Q5NUL3 1/20 0.41
GRM5 P41594 1/20 0.41
CYP2A6 P11509 1/20 0.39
EGLN1 Q9GZT9 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9495872 0.88 MCHR1 (0.52) MCHR1ACACBCHRM1HTR2ACYP2D6
SCHEMBL9855660 0.86 EGLN1 (0.48) MCHR1ACACBFFAR1FFAR4GRM5
SCHEMBL9494958 0.86 ACACB (0.49) MCHR1ACACBFFAR1FFAR4GRM5
SCHEMBL9498326 0.85 MCHR1 (0.55) MCHR1ACACBCHRM1HTR2ACYP2D6
SCHEMBL9497141 0.84 MCHR1 (0.54) MCHR1ACACBCHRM1HTR2ACYP2D6
SCHEMBL10520092 0.83 MCHR1 (0.46) MCHR1ACACBCHRM1CYP2D6FFAR1
SCHEMBL9500256 0.83 MCHR1 (0.53) MCHR1ACACBCHRM1HTR2AFFAR1
SCHEMBL9495546 0.83 ACACB (0.53) MCHR1ACACBCHRM1HTR2ACYP2D6
SCHEMBL9855141 0.82 FFAR1 (0.42) MCHR1ACACBFFAR1FFAR4CYP2A6
SCHEMBL9495802 0.82 ACACB (0.46) MCHR1ACACBFFAR1FFAR4GRM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0306505-B1 ACETYLENE DERIVATIVES AS COMPONENTS OF LIQUID CRYSTAL PHASES MERCK PATENT GmbH (DE) 1993-03-24 EP disclosed
US-5068053-A Liquid crystals for optical apparatus MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1991-11-26 US disclosed