SCHEMBL9499809

SCHEMBL9499809

CCOc1cnc(C#Cc2ccc([C@H]3CC[C@H](C)CC3)cc2)nc1

nearest known ligand 0.40

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ESR2 Q92731 1/20 0.40
ACACB O00763 11/20 0.37
MCHR1 Q99705 1/20 0.37
EGLN1 Q9GZT9 1/20 0.35
EGLN3 Q9H6Z9 1/20 0.35
HRH3 Q9Y5N1 1/20 0.35
MAOA P21397 1/20 0.34
MAOB P27338 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9499816 1.00 ESR2 (0.40) ESR2ACACBMCHR1EGLN1EGLN3
SCHEMBL10511453 0.94 MCHR1 (0.38) ESR2ACACBMCHR1HRH3MAOA
SCHEMBL9500347 0.90 MCHR1 (0.40) ESR2ACACBMCHR1HRH3MAOA
SCHEMBL9496182 0.90 ACACB (0.44) ACACBMCHR1EGLN1EGLN3MAOA
SCHEMBL9500360 0.90 MCHR1 (0.40) ESR2ACACBMCHR1HRH3MAOA
SCHEMBL9496173 0.90 ACACB (0.44) ACACBMCHR1EGLN1EGLN3MAOA
SCHEMBL9508530 0.89 ESR2 (0.46) ESR2ACACBHRH3MAOAMAOB
SCHEMBL5961794 0.89 ESR2 (0.46) ESR2ACACBHRH3MAOAMAOB
SCHEMBL9498316 0.89 RAB9A (0.46) ACACBMCHR1HRH3MAOAMAOB
SCHEMBL9498325 0.89 RAB9A (0.46) ACACBMCHR1HRH3MAOAMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0306505-B1 ACETYLENE DERIVATIVES AS COMPONENTS OF LIQUID CRYSTAL PHASES MERCK PATENT GmbH (DE) 1993-03-24 EP disclosed
US-5068053-A Liquid crystals for optical apparatus MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1991-11-26 US disclosed