SCHEMBL9501257

SCHEMBL9501257

Cc1cc(O)c(C)c(C)c1CC(NC(=O)OC(C)(C)C)C(=O)O

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACE P12821 2/20 0.49
ITGB3 P05106 2/20 0.44
ITGA2B P08514 2/20 0.44
CTSS P25774 4/20 0.43
PPARA Q07869 6/20 0.42
PPARG P37231 5/20 0.42
SCN9A Q15858 1/20 0.42
CTSK P43235 2/20 0.41
PTPN1 P18031 1/20 0.41
PPARD Q03181 2/20 0.41
CTSL P07711 1/20 0.40
CTSB P07858 1/20 0.40
ITGB1 P05556 1/20 0.40
ITGAV P06756 1/20 0.40
ITGB5 P18084 1/20 0.40
MAPT P10636 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
ALDH1A1 P00352 1/20 0.39
TSHR P16473 1/20 0.39
IDO1 P14902 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9304565 1.00 ACE (0.49) ACEITGB3ITGA2BCTSSPPARA
SCHEMBL1055585 0.86 ACE (0.52) ACEITGB3ITGA2BCTSSPPARA
SCHEMBL2263756 0.86 ACE (0.52) ACEITGB3ITGA2BCTSSPPARA
SCHEMBL10632461 0.85 ACE (0.49) ACEITGB3ITGA2BCTSSPPARA
SCHEMBL10632464 0.85 ACE (0.49) ACEITGB3ITGA2BCTSSPPARA
SCHEMBL2890189 0.84 ACE (0.53) ACEITGB3ITGA2BCTSSPPARA
SCHEMBL10604860 0.84 ACE (0.53) ACEITGB3ITGA2BCTSSPPARA
SCHEMBL7277748 0.82 ACE (0.51) ACEITGB3ITGA2BCTSSPPARA
SCHEMBL21062787 0.81 ACE (0.50) ACEITGB3ITGA2BCTSSPPARA
SCHEMBL9728451 0.81 ACE (0.50) ACEITGB3ITGA2BCTSSPPARA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5216124-A Analgesics G. D. SEARLE & CO. (US) 1993-06-01 US disclosed
US-5169833-A Analgesics G. D. SEARLE & CO. (US) 1992-12-08 US disclosed
US-4727189-A ANALGESICS, ANTIHYPERTENSIVE AGENTS G. D. SEARLE & CO. (US) 1988-02-23 US disclosed
US-4722922-A RENIN INHIBITION G. D. SEARLE & CO. (US) 1988-02-02 US disclosed
US-4603121-A ANALGESICS G. D. SEARLE & CO. (US) 1986-07-29 US disclosed
US-4599325-A ANALGESIC, HYPOTENSIVE G. D. SEARLE & CO. (US) 1986-07-08 US disclosed
EP-0154234-A2 Substituted tyrosil alanine dipeptide amides G.D. Searle & Co. (US) 1985-09-11 EP disclosed
EP-0136720-A2 Enkephalin analogs G.D. Searle & Co. (US) 1985-04-10 EP disclosed
US-4495178-A Enkephalin analogs G. D. SEARLE & CO. (US) 1985-01-22 US disclosed