SCHEMBL9501271

SCHEMBL9501271

C#CCN(Cc1ccc2nc(OC)[nH]c(=O)c2c1)c1ccc(C(=O)N[C@@H](CCC(=O)O)C(=O)O)cc1

nearest known ligand 0.82

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
TYMS P04818 12/20 0.82
DHFR P00374 1/20 0.72

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9223936 0.91 TYMS (0.68) TYMSDHFR
SCHEMBL9555830 0.90 TYMS (0.84) TYMSDHFR
SCHEMBL9556163 0.89 DHFR (0.73) TYMSDHFR
SCHEMBL9555871 0.89 TYMS (0.71) TYMSDHFR
SCHEMBL9501327 0.89 DHFR (0.91) TYMSDHFR
SCHEMBL9224063 0.89 DHFR (0.91) TYMSDHFR
SCHEMBL29363552 0.89 DHFR (0.91) TYMSDHFR
SCHEMBL29359823 0.89 DHFR (0.91) TYMSDHFR
SCHEMBL9556070 0.88 DHFR (0.72) TYMSDHFR
SCHEMBL9556172 0.88 TYMS (0.81) TYMSDHFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4992550-A Thymidylate synthetase inhibitors IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1991-02-12 US claimed
US-5252573-A Quinazoline derivatives IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1993-10-12 US disclosed
US-5187167-A Antitumor agents IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1993-02-16 US disclosed
US-5081124-A Amino acid and polyamino acid derivatives, inhibitors of thymidylate synthetase IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1992-01-14 US disclosed