SCHEMBL9501549

SCHEMBL9501549

COC=CC=C(C#N)C(=O)OC

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
APP P05067 2/20 0.48
ADORA2A P29274 1/20 0.38
ADORA2B P29275 1/20 0.38
ADORA1 P30542 1/20 0.38
KMT2A Q03164 7/20 0.36
MEN1 O00255 5/20 0.36
POLB P06746 3/20 0.36
KDM4E B2RXH2 5/20 0.35
MAPT P10636 8/20 0.34
LMNA P02545 6/20 0.34
ALDH1A1 P00352 4/20 0.34
TNNI3 P19429 1/20 0.34
CRHBP P24387 1/20 0.34
TNNT2 P45379 1/20 0.34
KLK7 P49862 1/20 0.34
TNNC1 P63316 1/20 0.34
CRHR2 Q13324 1/20 0.34
HTT P42858 1/20 0.33
GAA P10253 1/20 0.33
HPGD P15428 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9501545 1.00 APP (0.48) APPADORA2AADORA2BADORA1KMT2A
SCHEMBL21478208 0.82 APP (0.49) APPADORA2AADORA2BADORA1KMT2A
SCHEMBL28638384 0.82 CYP2C9 (0.54) KMT2AMEN1POLBKDM4EMAPT
SCHEMBL2396862 0.78 APP (0.52) APPADORA2AADORA2BADORA1KMT2A
SCHEMBL2396864 0.78 APP (0.52) APPADORA2AADORA2BADORA1KMT2A
SCHEMBL12292365 0.78 APP (0.52) APPADORA2AADORA2BADORA1KMT2A
SCHEMBL10488526 0.78 APP (0.37) APPKMT2AMEN1CYP2C9L3MBTL1
SCHEMBL18655709 0.77
SCHEMBL7618854 0.77
SCHEMBL7474650 0.77

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-55076863-A None JP disclosed
EP-0548291-A1 PYRIDYLTHIO OR PYRIDYLOXY ALKANOIC ACIDS SMITHKLINE BEECHAM CORPORATION (US) 1993-06-30 EP disclosed
WO-1992005156-A1 PYRIDYLTHIO OR PYRIDYLOXY ALKANOIC ACIDS SMITHKLINE BEECHAM CORPORATION (US) 1992-04-02 WO disclosed
US-4321387-A Process for the preparation of optically active nicotine analogs PHILIP MORRIS, INCORPORATED (US) 1982-03-23 US disclosed
JP-S5576863-A PREPARATION OF 2-CHLORONICOTINIC ACID YOSHITOMI PHARMACEUT IND LTD 1980-06-10 JP disclosed