SCHEMBL9501645

SCHEMBL9501645

CCOC(=O)C1=C(C)NC(C)=C(C(=O)OC)C1c1ccc(N)cc1

nearest known ligand 0.78

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 2/20 0.78
ALDH1A1 P00352 4/20 0.71
KDM4E B2RXH2 4/20 0.71
HSD17B10 Q99714 3/20 0.71
HPGD P15428 2/20 0.71
LMNA P02545 2/20 0.71
GAA P10253 1/20 0.71
TSHR P16473 4/20 0.70
SMN1; SMN2 Q16637 2/20 0.70
ABCC1 P33527 1/20 0.68
MEN1 O00255 3/20 0.64
KMT2A Q03164 3/20 0.64
POLB P06746 2/20 0.64
NPSR1 Q6W5P4 1/20 0.64
CACNA1F O60840 3/20 0.60
CACNA1D Q01668 3/20 0.60
CACNA1S Q13698 3/20 0.60
CACNA1C Q13936 3/20 0.60
HTT P42858 1/20 0.59
RAB9A P51151 1/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7817206 0.88 KDM4E (0.88) ADORA3ALDH1A1KDM4EHSD17B10HPGD
SCHEMBL3330194 0.88 ADORA3 (0.76) ADORA3ALDH1A1KDM4EHSD17B10HPGD
SCHEMBL20610477 0.87 ADORA3 (1.00) ADORA3ALDH1A1KDM4EHSD17B10HPGD
SCHEMBL7158354 0.86 ADORA3 (0.78) ADORA3ALDH1A1KDM4EHSD17B10HPGD
SCHEMBL14576820 0.85 ADORA3 (0.68) ADORA3ALDH1A1KDM4EHSD17B10HPGD
SCHEMBL11835842 0.85 ADORA3 (0.72) ADORA3ALDH1A1KDM4EHSD17B10HPGD
SCHEMBL8288455 0.84 ADORA3 (0.74) ADORA3ALDH1A1KDM4EHSD17B10HPGD
SCHEMBL7163210 0.84 ADORA3 (0.70) ADORA3ALDH1A1KDM4EHSD17B10HPGD
SCHEMBL3032293 0.84 KDM4E (0.80) ADORA3ALDH1A1KDM4EHSD17B10HPGD
SCHEMBL7159073 0.83 ADORA3 (1.00) ADORA3ALDH1A1KDM4EHSD17B10HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0458823-B1 A PROCESS FOR PREPARATION OF ENANTIOMERICALLY PURE POLYSUBSTITUTED 1,4-DIHYDROPYRIDINES BOEHRINGER MANNHEIM ITALIA S.P.A. (IT) 1993-10-13 EP disclosed
US-5245039-A PROCESS FOR PREPARATION OF ENANTIOMERICALLY PURE POLYSUBSTITUTED 1,4-DIHYDROPYRIDINES BOEHRINGER MANNHEIM ITALIA (IT) 1993-09-14 US disclosed
EP-0458823-A1 A PROCESS FOR PREPARATION OF ENANTIOMERICALLY PURE POLYSUBSTITUTED 1,4-DIHYDROPYRIDINES. BOEHRINGER MANNHEIM ITALIA (IT) 1991-12-04 EP disclosed
WO-1990009376-A1 A PROCESS FOR PREPARATION OF ENANTIOMERICALLY PURE POLYSUBSTITUTED 1,4-DIHYDROPYRIDINES BOEHRINGER MANNHEIM ITALIA S.P.A. (IT) 1990-08-23 WO disclosed
EP-0383320-A1 A process for preparation of enantiomerically pure polysubstituted 1,4-dihydropyridines BOEHRINGER MANNHEIM ITALIA S.P.A. (IT) 1990-08-22 EP disclosed