SCHEMBL9503104

SCHEMBL9503104

CC(=O)NCCSC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCC1CN=C(c2ccccc2F)c2ccccc2N1C

nearest known ligand 0.87

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CCKBR P32239 9/20 0.66
OPRD1 P41143 2/20 0.49
OPRK1 P41145 2/20 0.49
CCKAR P32238 2/20 0.45
OPRM1 P35372 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9528505 0.93 CCKBR (0.67) CCKBROPRD1OPRK1CCKAR
Water SCHEMBL10666524 0.92 CCKBR (0.66) CCKBROPRD1OPRK1CCKAR
SCHEMBL9501387 0.79 CCKBR (1.00) CCKBROPRD1OPRK1CCKAR
SCHEMBL9503082 0.78 CCKBR (0.53) CCKBROPRD1OPRK1CCKAROPRM1
SCHEMBL10868746 0.75 CCKBR (0.68) CCKBROPRD1OPRK1OPRM1
SCHEMBL9499260 0.74 CCKBR (1.00) CCKBROPRD1OPRK1OPRM1
Water SCHEMBL9503005 0.74 CCKBR (0.98) CCKBROPRD1OPRK1OPRM1
SCHEMBL9501135 0.72 CCKBR (0.64) CCKBROPRD1OPRK1OPRM1
SCHEMBL10803682 0.70 CCKBR (0.75) CCKBROPRD1OPRK1OPRM1
SCHEMBL9529624 0.70 CCKBR (0.69) CCKBROPRD1OPRK1OPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5206238-A Cholecystokinin antagonists MERCK & CO., INC. (US) 1993-04-27 US disclosed