SCHEMBL9503479

SCHEMBL9503479

CS(=O)(=O)Nc1ccccc1OC1CCCCC1O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MRGPRX1 Q96LB2 1/20 0.43
CYP19A1 P11511 3/20 0.43
PTGS1 P23219 6/20 0.42
PTGS2 P35354 5/20 0.42
ALDH1A1 P00352 5/20 0.42
KMT2A Q03164 3/20 0.42
SMN1; SMN2 Q16637 3/20 0.42
MEN1 O00255 2/20 0.42
TSHR P16473 2/20 0.42
PTGES O14684 1/20 0.42
CYP1A2 P05177 1/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2D6 P10635 1/20 0.42
MAPT P10636 1/20 0.42
ALOX15 P16050 1/20 0.42
CYP2C19 P33261 1/20 0.42
NPY1R P25929 1/20 0.40
NPY2R P49146 1/20 0.40
NPY4R P50391 1/20 0.40
NPY5R Q15761 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8523784 0.80 PTGS1 (0.61) MRGPRX1CYP19A1PTGS1PTGS2ALDH1A1
SCHEMBL9502723 0.78 CYP19A1 (0.73) CYP19A1PTGS1PTGS2ALDH1A1KMT2A
SCHEMBL9511659 0.77 MRGPRX1 (0.47) MRGPRX1CYP19A1PTGS1PTGS2ALDH1A1
SCHEMBL20022642 0.77 NPY1R (0.50) ALDH1A1KMT2ASMN1; SMN2MEN1TSHR
SCHEMBL9501603 0.76 PTGS2 (0.43) MRGPRX1CYP19A1PTGS1PTGS2ALDH1A1
SCHEMBL1496601 0.73 NPY1R (0.47) ALDH1A1KMT2AMEN1CYP2D6NPY1R
SCHEMBL9501963 0.72 CYP19A1 (0.47) MRGPRX1CYP19A1PTGS1PTGS2ALDH1A1
SCHEMBL1496734 0.72 NPY1R (0.46) KMT2AMEN1NPY1RNPY2RNPY4R
SCHEMBL6378390 0.70 PTGS1 (0.56) CYP19A1PTGS1PTGS2ALDH1A1KMT2A
SCHEMBL1496646 0.70 NPY1R (0.44) ALDH1A1KMT2AMEN1CYP2D6NPY1R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0317332-B1 SULFONANILIDE COMPOUNDS TAISHO PHARMACEUTICAL CO. LTD (JP) 1993-05-19 EP disclosed
US-4885367-A ANTIINFLAMMATORY AGENTS, ANTIPYRETICS, ANALGESICS; SIDE EFFECT REDUCTION TAISHO PHARMACEUTICAL CO., LTD. (JP) 1989-12-05 US disclosed
EP-0317332-A2 Sulfonanilide compounds TAISHO PHARMACEUTICAL CO. LTD (JP) 1989-05-24 EP disclosed