SCHEMBL9504546

SCHEMBL9504546

CCCn1c(=O)[nH]c(=O)c2c1ncn2Cc1ccc(OC)cc1

nearest known ligand 0.66

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 4/20 0.66
ADORA2A P29274 4/20 0.66
PDE4B Q07343 4/20 0.66
PDE4C Q08493 4/20 0.66
PDE4D Q08499 4/20 0.66
BRD4 O60885 9/20 0.60
BRD2 P25440 2/20 0.57
BRD3 Q15059 2/20 0.57
BRDT Q58F21 2/20 0.57
ALDH1A1 P00352 3/20 0.57
MEN1 O00255 2/20 0.57
KMT2A Q03164 2/20 0.57
KDM4E B2RXH2 2/20 0.50
HPGD P15428 2/20 0.50
NPSR1 Q6W5P4 1/20 0.50
GAA P10253 1/20 0.48
MAPT P10636 1/20 0.48
HTT P42858 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL555712 0.88 BRD4 (0.71) BRD4BRD2BRD3BRDTALDH1A1
SCHEMBL7607643 0.87 PDE4A (0.74) PDE4AADORA2APDE4BPDE4CPDE4D
SCHEMBL12687220 0.86 KDM4E (0.56) BRD4BRD2BRD3BRDTALDH1A1
SCHEMBL3104007 0.81 MEN1 (0.75) PDE4AADORA2APDE4BPDE4CPDE4D
SCHEMBL3902928 0.80 PDE4A (1.00) PDE4AADORA2APDE4BPDE4CPDE4D
SCHEMBL1713302 0.80 MEN1 (0.70) PDE4AADORA2APDE4BPDE4CPDE4D
SCHEMBL556875 0.80 BRD4 (0.65) PDE4AADORA2APDE4BPDE4CPDE4D
SCHEMBL21381257 0.79 PDE4A (1.00) PDE4AADORA2APDE4BPDE4CPDE4D
SCHEMBL9842832 0.79 BRD4 (0.50) ADORA2ABRD4BRD2BRD3BRDT
SCHEMBL557088 0.79 MEN1 (0.68) PDE4AADORA2APDE4BPDE4CPDE4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-5001065-A None JP disclosed
JP-3167186-A None JP disclosed
JP-H051065-A XANTHINE DERIVATIVE HOKURIKU SEIYAKU CO LTD 1993-01-08 JP disclosed
JP-H03167186-A XANTHINE DERIVATIVE AND USE THEREOF HOKURIKU SEIYAKU CO LTD 1991-07-19 JP disclosed