SCHEMBL9842832

SCHEMBL9842832

COc1ccc(Cn2cnc3c2c(=O)[nH]c(=O)n3C2CC2)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 4/20 0.50
OPRM1 P35372 1/20 0.49
TPH1 P17752 2/20 0.48
TPH2 Q8IWU9 2/20 0.48
BRD2 P25440 1/20 0.46
BRD3 Q15059 1/20 0.46
BRDT Q58F21 1/20 0.46
DRD2 P14416 1/20 0.45
DRD4 P21917 1/20 0.45
DRD3 P35462 1/20 0.45
HPGD P15428 3/20 0.43
KDM4E B2RXH2 2/20 0.43
ALDH1A1 P00352 2/20 0.43
MAPT P10636 2/20 0.43
HTT P42858 2/20 0.43
GAA P10253 1/20 0.43
CYP11B2 P19099 1/20 0.43
NPSR1 Q6W5P4 1/20 0.42
TP53 P04637 1/20 0.41
ADORA2A P29274 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7603126 0.85 BRD4 (0.58) BRD4OPRM1TPH1TPH2BRD2
SCHEMBL12687220 0.83 KDM4E (0.56) BRD4BRD2BRD3BRDTHPGD
SCHEMBL555712 0.80 BRD4 (0.71) BRD4BRD2BRD3BRDTHPGD
SCHEMBL9504546 0.79 PDE4A (0.66) BRD4BRD2BRD3BRDTHPGD
SCHEMBL9842744 0.79 PDE5A (0.50) KDM4EMAPTCYP11B2TP53ADORA2A
SCHEMBL9842568 0.79 PDE4A (0.59) BRD4BRD2BRD3BRDTKDM4E
SCHEMBL7464187 0.77 PDE4A (0.65) BRD4BRD2BRD3BRDTKDM4E
SCHEMBL9842833 0.75 ALDH1A1 (0.67) BRD4BRD2BRD3BRDTHPGD
SCHEMBL9615238 0.75 SMN1; SMN2 (0.44) BRD4BRD2BRD3BRDTKDM4E
SCHEMBL9842911 0.74 MEN1 (0.62) BRD4BRD2BRD3BRDTKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0430025-A2 Xanthine compound, method for preparing thereof, and a pharmaceutical composition comprising the same HOKURIKU PHARMACEUTICAL CO., LTD. (JP) 1991-06-05 EP disclosed