SCHEMBL950478

SCHEMBL950478

COCOc1cccc(C=O)c1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.60
RAB9A P51151 2/20 0.60
TDP1 Q9NUW8 1/20 0.60
MAOA P21397 7/20 0.58
MAOB P27338 7/20 0.58
SRC P12931 1/20 0.49
ALDH1A1 P00352 3/20 0.44
POLB P06746 1/20 0.44
KDM4E B2RXH2 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
CCNB2 O95067 2/20 0.42
CDK1 P06493 2/20 0.42
CDK4 P11802 2/20 0.42
CCNB1 P14635 2/20 0.42
CCND1 P24385 2/20 0.42
CCNB3 Q8WWL7 2/20 0.42
TTR P02766 1/20 0.41
FDPS P14324 1/20 0.41
CHRM2 P08172 1/20 0.41
CHRM1 P11229 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29955275 1.00 NPC1 (0.60) NPC1RAB9ATDP1MAOAMAOB
SCHEMBL10800526 0.92 NPC1 (0.54) NPC1RAB9ATDP1MAOAMAOB
SCHEMBL5001878 0.85 NPC1 (0.54) NPC1RAB9ATDP1MAOAMAOB
SCHEMBL30855377 0.84 NPC1 (0.59) NPC1RAB9ATDP1MAOAMAOB
SCHEMBL1279355 0.84 NPC1 (0.59) NPC1RAB9ATDP1MAOAMAOB
SCHEMBL8709017 0.83 CCNB2 (0.62) NPC1RAB9ATDP1MAOAMAOB
SCHEMBL8709013 0.83 CCNB2 (0.62) NPC1RAB9ATDP1MAOAMAOB
SCHEMBL8111540 0.83 MAOA (0.55) NPC1RAB9ATDP1MAOAMAOB
SCHEMBL30833931 0.83 MAOA (0.55) NPC1RAB9ATDP1MAOAMAOB
SCHEMBL695627 0.83 NPC1 (0.57) NPC1RAB9ATDP1MAOAMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 133 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112826812-B Pharmaceutical composition for treating colon cancer and application thereof 青岛大学 2023-08-25 CN disclosed
CN-112694392-B TRPV3 inhibitor and preparation method thereof 青岛大学 2022-11-22 CN disclosed
CN-114591267-A Nitrogen-containing derivatives of monocarbonyl curcumin, and preparation method and application thereof 沈阳药科大学 2022-06-07 CN disclosed
CN-112826812-A Pharmaceutical composition for treating colon cancer and application thereof 青岛大学 2021-05-25 CN disclosed
CN-112694392-A TRPV3 inhibitor and preparation method thereof 青岛大学 2021-04-23 CN disclosed
EP-2883865-B1 Compound capable of binding S1P receptor and pharmaceutical use thereof ONO PHARMACEUTICAL CO (JP) 2019-09-25 EP disclosed
US-9884836-B2 2-substituted-5-hydroxy-4H-chromen-4-ones as novel ligands for the serotonin receptor 2B (5-HT2B) VIRGINIA COMMONWEALTH UNIVERSITY (US) 2018-02-06 US disclosed
EP-3150203-A1 COMPOUNDS WITH (1E,6E)-1,7-BIS-(3,4- DIMETHOXYPHENYL)-4,4-DISSTITUTED-HEPA-1,6-DIENE-3,5-DI-ONE STRUCTURAL SCAFFOLD,THEIR BIOLOGICAL ACTIVITY, AND USES THEREOF Allianz Pharmascience Ltd (TW) 2017-04-05 EP disclosed
EP-1926737-B1 4-AMINO-THIENO[3,2-C]PYRIDINE-7-CARBOXYLIC ACID DERIVATIVES HOFFMANN LA ROCHE (CH) 2017-03-15 EP disclosed
US-9562025-B2 Compounds with (1E, 6E)-1,7-Bis-(3,4-dimethoxyphenyl)-4-4-distributed-hepta-1,6-diene-3,5-dione structural scaffold, their biological activity, and uses thereof ALLIANZ PHARMASCIENCE LTD. (TW) 2017-02-07 US disclosed
EP-0262870-A2 Morpholine, piperidine and tetrahydropyridine derivatives, processes for their preparation and their use as fungicides SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1988-04-06 EP disclosed
US-4220767-A HISTAMINE ANTAGONISTS SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1980-09-02 US disclosed
US-4185103-A ANTAGONISTS SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1980-01-22 US disclosed
US-4155935-A Benzylamine analgesics AMERICAN HOME PRODUCTS CORPORATION (US) 1979-05-22 US disclosed
US-4125530-A FROM 1,1-DIHALO-3,3,3-TRIFLUOROACETONE, BASE, AMMONIA AND A CARBOXALDEHYDE MERCK & CO., INC. (US) 1978-11-14 US disclosed
US-4032522-A ANTI-GOUT, ANTI-HYPERURICEMIC MERCK & CO., INC. (US) 1977-06-28 US disclosed
US-4017637-A Benzylamine analgesics AMERICAN HOME PRODUCTS CORPORATION (US) 1977-04-12 US disclosed
US-3987105-A PROCESS FOR METHOXYMETHYLATION OF PHENOLIC HYDROXYL GROUPS AMERICAN HOME PRODUCTS CORPORATION (US) 1976-10-19 US disclosed
US-3975436-A Benzylamine narcotic antagonists AMERICAN HOME PRODUCTS CORPORATION (US) 1976-08-17 US disclosed
US-3937818-A ADMINISTERING AMERICAN HOME PRODUCTS CORPORATION (US) 1976-02-10 US disclosed