SCHEMBL951110

SCHEMBL951110

Cc1cn(-c2ccc(C#N)cc2)c2cccc(-c3cnc4ccccc4c3)c12

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 13/20 0.53
PTGS1 P23219 1/20 0.39
PTGS2 P35354 1/20 0.39
PIK3CA P42336 3/20 0.38
MTOR P42345 3/20 0.38
PIK3C2A O00443 2/20 0.38
PIK3C2B O00750 2/20 0.38
PIK3CD O00329 2/20 0.38
PIK3CB P42338 2/20 0.38
PIK3CG P48736 2/20 0.38
PRKDC P78527 2/20 0.38
ATM Q13315 2/20 0.38
CHEK1 O14757 1/20 0.38
ABCB11 O95342 1/20 0.38
CSF1R P07333 1/20 0.38
MET P08581 1/20 0.38
PIK3R1 P27986 1/20 0.38
LTK P29376 1/20 0.38
CDK7 P50613 1/20 0.38
NEK2 P51955 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL952602 0.85 HSP90AA1 (0.51) HSP90AA1PTGS1PTGS2PIK3CAMTOR
SCHEMBL951144 0.83 HSP90AA1 (0.65) HSP90AA1
SCHEMBL421583 0.82 HSP90AA1 (0.53) HSP90AA1PIK3CAMTORPIK3C2APIK3C2B
SCHEMBL950332 0.80 HSP90AA1 (0.51) HSP90AA1PTGS1PTGS2PIK3CAMTOR
SCHEMBL947823 0.78 PIK3CA (0.40) HSP90AA1PTGS1PTGS2PIK3CAMTOR
SCHEMBL949997 0.77 HSP90AA1 (0.75) HSP90AA1
SCHEMBL421857 0.76 HSP90AA1 (0.51) HSP90AA1PIK3CAMTORPIK3C2APIK3C2B
SCHEMBL2692049 0.71 HSP90AA1 (0.54) HSP90AA1
SCHEMBL15445880 0.70 PDGFRB (0.60) PIK3CAMTORPIK3CDPIK3CBPIK3CG
SCHEMBL12944196 0.70 HSP90AA1 (0.87) HSP90AA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011004132-A1 NOVEL HSP90-INHIBITING INDOLE DERIVATIVES, COMPOSITIONS CONTAINING SAID DERIVATIVES, AND USE THEREOF SANOFI-AVENTIS (FR) 2011-01-13 WO disclosed