SCHEMBL950332

SCHEMBL950332

N#Cc1ccc(-n2ccc3c(-c4cnc5ccccc5c4)cccc32)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 2/20 0.51
CYP19A1 P11511 1/20 0.42
PDGFRB P09619 2/20 0.39
PDGFRA P16234 2/20 0.39
PIK3CA P42336 3/20 0.37
MTOR P42345 3/20 0.37
PIK3C2A O00443 2/20 0.37
PIK3C2B O00750 2/20 0.37
PIK3CD O00329 2/20 0.37
PIK3CB P42338 2/20 0.37
PIK3CG P48736 2/20 0.37
PRKDC P78527 2/20 0.37
ATM Q13315 2/20 0.37
MET P08581 2/20 0.37
CHEK1 O14757 1/20 0.37
ABCB11 O95342 1/20 0.37
CSF1R P07333 1/20 0.37
PIK3R1 P27986 1/20 0.37
LTK P29376 1/20 0.37
CDK7 P50613 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL950675 0.85 HSP90AA1 (0.49) HSP90AA1CYP19A1PDGFRBPDGFRAPIK3CA
SCHEMBL421857 0.83 HSP90AA1 (0.51) HSP90AA1PDGFRBPDGFRAPIK3CAMTOR
SCHEMBL951469 0.81 HSP90AA1 (0.62) HSP90AA1CLK4MAP4K5
SCHEMBL947823 0.81 PIK3CA (0.40) HSP90AA1PDGFRBPDGFRAPIK3CAMTOR
SCHEMBL951110 0.80 HSP90AA1 (0.53) HSP90AA1PIK3CAMTORPIK3C2APIK3C2B
SCHEMBL421583 0.76 HSP90AA1 (0.53) HSP90AA1PIK3CAMTORPIK3C2APIK3C2B
SCHEMBL22064668 0.73 BIRC5 (0.45) PDGFRBPDGFRAPIK3CAMTORPIK3CD
SCHEMBL15445880 0.73 PDGFRB (0.60) PDGFRBPDGFRAPIK3CAMTORPIK3CD
SCHEMBL420055 0.70 HSP90AA1 (0.49) HSP90AA1PDGFRBPDGFRAPIK3CAMTOR
SCHEMBL2198777 0.70 PDGFRB (0.60) HSP90AA1PDGFRBPDGFRAPIK3CAMTOR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011004132-A1 NOVEL HSP90-INHIBITING INDOLE DERIVATIVES, COMPOSITIONS CONTAINING SAID DERIVATIVES, AND USE THEREOF SANOFI-AVENTIS (FR) 2011-01-13 WO disclosed