SCHEMBL9511765

SCHEMBL9511765

BrCCCCCCOCCc1cc2ccccc2s1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AGXT P21549 1/20 0.45
CYP2A6 P11509 3/20 0.45
ASIC3 Q9UHC3 1/20 0.45
LOXL2 Q9Y4K0 1/20 0.45
ADRB2 P07550 1/20 0.42
CHRNA7 P36544 1/20 0.38
GLS O94925 1/20 0.38
ADRA1D P25100 2/20 0.36
IDH1 O75874 1/20 0.35
HDAC3 O15379 1/20 0.34
HDAC4 P56524 1/20 0.34
HDAC1 Q13547 1/20 0.34
HDAC7 Q8WUI4 1/20 0.34
HDAC2 Q92769 1/20 0.34
HDAC10 Q969S8 1/20 0.34
HDAC11 Q96DB2 1/20 0.34
HDAC8 Q9BY41 1/20 0.34
HDAC6 Q9UBN7 1/20 0.34
HDAC9 Q9UKV0 1/20 0.34
HDAC5 Q9UQL6 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9587702 0.85 CYP2A6 (0.53) AGXTCYP2A6ASIC3LOXL2ADRB2
SCHEMBL48281 0.82 CYP2A6 (0.56) AGXTCYP2A6ASIC3LOXL2ADRB2
SCHEMBL48175 0.82 AGXT (0.47) AGXTCYP2A6ASIC3LOXL2ADRB2
SCHEMBL4283571 0.81 CYP2A6 (0.56) AGXTCYP2A6ASIC3LOXL2ADRB2
SCHEMBL2089869 0.78 AGXT (0.46) AGXTCYP2A6ASIC3LOXL2ADRB2
SCHEMBL4047968 0.78 CYP2A6 (0.60) AGXTCYP2A6ASIC3LOXL2ADRB2
SCHEMBL2095290 0.75 AGXT (0.49) AGXTCYP2A6ASIC3LOXL2ADRB2
SCHEMBL9510811 0.74 AGXT (0.45) AGXTLOXL2GLSHDAC3HDAC4
SCHEMBL9510780 0.74 AGXT (0.45) AGXTLOXL2GLSHDAC3HDAC4
SCHEMBL2095661 0.73 CYP2A6 (0.55) AGXTCYP2A6ASIC3LOXL2ADRB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0322164-B1 ETHANOLAMINE DERIVATIVES GLAXO GROUP LIMITED (GB) 1993-09-22 EP disclosed
US-5039697-A Adrenergic stimulants, bronchodilators GLAXO GROUP LIMITED (GB) 1991-08-13 US disclosed
US-5032609-A Ethanolamine derivatives GLAXO GROUP LIMITED (GB) 1991-07-16 US disclosed
US-5002966-A Adrenergic Stimulants GLAXO GROUP LIMITED (GB) 1991-03-26 US disclosed
EP-0322164-A2 Ethanolamine derivatives GLAXO GROUP LIMITED (GB) 1989-06-28 EP disclosed