SCHEMBL9587702

SCHEMBL9587702

BrCCCCCCc1cc2ccccc2s1

nearest known ligand 0.53

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 4/20 0.53
ASIC3 Q9UHC3 1/20 0.53
LOXL2 Q9Y4K0 1/20 0.53
AGXT P21549 1/20 0.49
ADRB2 P07550 1/20 0.49
GLS O94925 2/20 0.45
ADRA1D P25100 2/20 0.41
IDH1 O75874 1/20 0.40
CTRC Q99895 1/20 0.38
MGLL Q99685 1/20 0.37
CHRNA7 P36544 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4283571 0.93 CYP2A6 (0.56) CYP2A6ASIC3LOXL2AGXTADRB2
SCHEMBL4047968 0.85 CYP2A6 (0.60) CYP2A6ASIC3LOXL2AGXTADRB2
SCHEMBL9511765 0.85 AGXT (0.45) CYP2A6ASIC3LOXL2AGXTADRB2
SCHEMBL24614167 0.83 CYP2A6 (0.53) CYP2A6ASIC3LOXL2AGXTADRB2
SCHEMBL9347724 0.83 CYP2A6 (0.53) CYP2A6ASIC3LOXL2AGXTADRB2
SCHEMBL1687607 0.83 CYP2A6 (0.53) CYP2A6ASIC3LOXL2AGXTADRB2
SCHEMBL2091527 0.83 CYP2A6 (0.53) CYP2A6ASIC3LOXL2AGXTADRB2
SCHEMBL9347774 0.83 CYP2A6 (0.53) CYP2A6ASIC3LOXL2AGXTADRB2
SCHEMBL9672464 0.82 CYP2A6 (0.49) CYP2A6ASIC3LOXL2AGXTADRB2
SCHEMBL30665226 0.81 CYP2A6 (0.64) CYP2A6ASIC3LOXL2AGXTADRB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5258400-A Immunosuppressive compounds for psoriasis ALLERGAN, INC. (US) 1993-11-02 US disclosed
EP-0295056-B1 ANTI-INFLAMMATORY FURANONES ALLERGAN, INC (US) 1992-08-05 EP disclosed
US-5134128-A Immunosuppressive and antiproliferative activity for psoriasis and calcium homeostasis ALLERGAN, INC. (US) 1992-07-28 US disclosed
US-5112853-A Antiarthritic, calcium channel blockers, immunosuppresive ALLERGAN, INC. (US) 1992-05-12 US disclosed
EP-0429287-A2 Anti-inflammatory furanone compounds ALLERGAN, INC. (US) 1991-05-29 EP disclosed
EP-0295056-A1 Anti-inflammatory furanones ALLERGAN, INC (US) 1988-12-14 EP disclosed