SCHEMBL9513526

SCHEMBL9513526

CNC(=S)N1CCN(C=O)CC1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.45
MAPT P10636 3/20 0.45
LMNA P02545 1/20 0.45
NPSR1 Q6W5P4 1/20 0.43
POLB P06746 4/20 0.42
RECQL P46063 1/20 0.42
KDM4E B2RXH2 1/20 0.42
CYP1A2 P05177 2/20 0.41
CYP3A4 P08684 2/20 0.41
CYP2C9 P11712 2/20 0.41
CYP2C19 P33261 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
PKM P14618 1/20 0.40
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
HTT P42858 1/20 0.39
RAB9A P51151 3/20 0.38
NPC1 O15118 2/20 0.38
TDP1 Q9NUW8 1/20 0.38
TSHR P16473 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11284619 0.82
SCHEMBL7663156 0.77 POLB (0.70) ALDH1A1MAPTPOLBRECQLKMT2A
SCHEMBL14289057 0.75 POLB (0.38) ALDH1A1MAPTNPSR1POLBRECQL
SCHEMBL11531296 0.73 MGLL (0.50) ALDH1A1MAPTLMNAPOLBRECQL
SCHEMBL11528813 0.72
SCHEMBL14289031 0.72 POLB (0.35) ALDH1A1MAPTNPSR1POLBRECQL
SCHEMBL5092718 0.71 TSHR (0.38) NPSR1RECQLKMT2ARAB9ATSHR
SCHEMBL11530138 0.70 NPC1 (0.47) ALDH1A1MAPTPOLBRECQLKDM4E
SCHEMBL10448785 0.70 NPC1 (0.47) ALDH1A1MAPTPOLBRECQLKDM4E
SCHEMBL1307070 0.69 CYP1A2 (0.54) ALDH1A1KDM4ECYP1A2SMN1; SMN2KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0233051-B1 ANTIARRHYTHMIC AGENTS Pfizer Limited (GB) 1993-09-15 EP disclosed
US-4806536-A Piperazinyl-substituted pyridine and imidazole anti-arrhythmic agents PFIZER, INC. (US) 1989-02-21 US disclosed
EP-0233051-A2 Antiarrhythmic Agents Pfizer Limited (GB) 1987-08-19 EP disclosed