SCHEMBL9514129

SCHEMBL9514129

O=[N+]([O-])CCc1ccc2ccccc2c1

nearest known ligand 0.49

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.49
CYP2A6 P11509 1/20 0.47
SIGMAR1 Q99720 2/20 0.46
HRH3 Q9Y5N1 1/20 0.45
KMT2A Q03164 2/20 0.43
MEN1 O00255 1/20 0.43
MAPT P10636 1/20 0.43
ALPG P10696 1/20 0.43
HDAC1 Q13547 1/20 0.43
HDAC8 Q9BY41 1/20 0.43
TLR4 O00206 1/20 0.43
TLR2 O60603 1/20 0.43
NR1D1 P20393 1/20 0.42
SLC13A5 Q86YT5 1/20 0.42
PDPK1 O15530 1/20 0.42
SLC6A4 P31645 1/20 0.41
CNR1 P21554 1/20 0.41
CNR2 P34972 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6644343 0.81 CYP1A2 (0.50) CYP1A2CYP2A6SIGMAR1KMT2AMEN1
SCHEMBL9423246 0.79 MAPT (0.55) CYP1A2KMT2AMEN1MAPTALPG
SCHEMBL188307 0.78 TSHR (0.42) CYP1A2SIGMAR1KMT2AMEN1CNR1
SCHEMBL17541809 0.77 TSHR (0.46) CYP1A2SIGMAR1HRH3CNR1
SCHEMBL29560700 0.77 CYP1A2 (0.65) CYP1A2CYP2A6SIGMAR1HRH3KMT2A
SCHEMBL6240981 0.77 CYP1A2 (0.65) CYP1A2CYP2A6SIGMAR1HRH3KMT2A
SCHEMBL264237 0.76 CNR1 (0.46) CYP1A2CYP2A6SIGMAR1CNR1
Hydrogen Peroxide SCHEMBL28697848 0.74 CYP1A2 (0.47) CYP1A2SIGMAR1HDAC1HDAC8CNR1
SCHEMBL131160 0.74 CYP1A2 (0.56) CYP1A2CYP2A6SIGMAR1HRH3HDAC1
SCHEMBL29213229 0.74 MAPK1 (0.54) CYP1A2KMT2AMEN1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1022319-C 1, 2, 3, 4-tetrahydronaphthalene derivatives, process for their preparation and their use as medicaments MERRELL DOW PHARMA (US) 1993-10-06 CN disclosed
EP-0378456-B1 TETRALIN DERIVATIVES MERRELL DOW PHARMACEUTICALS INC. (US) 1993-09-15 EP disclosed
US-5106861-A Method of using certain tetralin derivatives to produce analgesic relief MERRELL DOW PHARMACEUTICALS INC. (US) 1992-04-21 US disclosed
US-5041673-A Aminopeptidase inhibitors, immunomodulators, analgesics MERRELL DOW PHARMACEUTICALS INC. (US) 1991-08-20 US disclosed
EP-0381902-A1 Tetralin derivatives MERRELL DOW PHARMACEUTICALS INC. (US) 1990-08-16 EP disclosed
CN-1044460-A Novel 1,2,3,4-tetralin derivative MERRELL DOW PHARMA (US) 1990-08-08 CN disclosed
EP-0378456-A1 Tetralin derivatives MERRELL DOW PHARMACEUTICALS INC. (US) 1990-07-18 EP disclosed