SCHEMBL9515044

SCHEMBL9515044

CCOC(=O)/C(=C(\C)N)C(c1cccc(C(F)(F)F)c1)C(C(=O)CCl)C(=O)OCC

nearest known ligand 0.41

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
EPHX1 P07099 3/20 0.41
GAA P10253 4/20 0.40
MAPT P10636 2/20 0.40
ALOX12 P18054 2/20 0.40
ATM Q13315 2/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
HPGD P15428 2/20 0.39
ALDH1A1 P00352 1/20 0.39
PNMT P11086 1/20 0.38
XPO1 O14980 1/20 0.37
PPARG P37231 2/20 0.36
SLC22A12 Q96S37 1/20 0.36
THRB P10828 1/20 0.36
CHRM2 P08172 1/20 0.36
CHRM4 P08173 1/20 0.36
CHRM3 P20309 1/20 0.36
CES2 O00748 1/20 0.36
GPR35 Q9HC97 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9515054 1.00 EPHX1 (0.41) EPHX1GAAMAPTALOX12ATM
SCHEMBL9514242 0.94 GAA (0.41) EPHX1GAAMAPTALOX12ATM
SCHEMBL9514236 0.94 GAA (0.41) EPHX1GAAMAPTALOX12ATM
SCHEMBL9515045 0.86 GAA (0.38) GAAMAPTSMN1; SMN2ALDH1A1XPO1
SCHEMBL9515051 0.86 GAA (0.38) GAAMAPTSMN1; SMN2ALDH1A1XPO1
SCHEMBL9511451 0.80 SMN1; SMN2 (0.43) GAAMAPTALOX12ATMSMN1; SMN2
SCHEMBL21399776 0.79 EPHX1 (0.49) EPHX1GAAMAPTALOX12ATM
SCHEMBL21382300 0.79 EPHX1 (0.53) EPHX1GAAMAPTALOX12ATM
SCHEMBL9512935 0.77 GAA (0.43) GAAMAPTHPGDALDH1A1
SCHEMBL9512946 0.77 GAA (0.43) GAAMAPTHPGDALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0212340-B1 2-(heteroalkyl)-1,4-dihydropyridines, process for their preparations and pharmaceutical compositions containing them BOEHRINGER MANNHEIM ITALIA (IT) 1993-10-27 EP disclosed
US-4839348-A HYPOTENSIVE AGENTS; ANTICOAGULANTS, ANTIISCHEMIC AGENTS BOEHRINGER BIOCHEMIA ROBIN S.P.A. (IT) 1989-06-13 US disclosed
EP-0212340-A1 2-(heteroalkyl)-1,4-dihydropyridines, process for their preparations and pharmaceutical compositions containing them BOEHRINGER MANNHEIM ITALIA S.P.A. (IT) 1987-03-04 EP disclosed