SCHEMBL9512946

SCHEMBL9512946

CCOC(=O)C(=C(C)N)C(c1cccc([N+](=O)[O-])c1)C(C(=O)CCl)C(=O)OC

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.43
GLO1 Q04760 1/20 0.43
LMNA P02545 5/20 0.42
KMT2A Q03164 5/20 0.42
ALDH1A1 P00352 5/20 0.42
KDM4E B2RXH2 1/20 0.42
CYP3A4 P08684 4/20 0.41
CYP2C9 P11712 4/20 0.41
CYP2C19 P33261 4/20 0.41
CYP2D6 P10635 3/20 0.41
NPSR1 Q6W5P4 3/20 0.41
MAPT P10636 5/20 0.40
HIF1A Q16665 3/20 0.40
CYP1A2 P05177 3/20 0.40
MEN1 O00255 3/20 0.40
TSHR P16473 2/20 0.40
NFKB1 P19838 2/20 0.40
MAPK1 P28482 2/20 0.40
POLB P06746 1/20 0.40
GPR55 Q9Y2T6 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9512935 1.00 GAA (0.43) GAAGLO1LMNAKMT2AALDH1A1
SCHEMBL9515051 0.79 GAA (0.38) GAAKMT2AALDH1A1NPSR1MAPT
SCHEMBL9515045 0.79 GAA (0.38) GAAKMT2AALDH1A1NPSR1MAPT
SCHEMBL9515044 0.77 EPHX1 (0.41) GAAALDH1A1MAPTHPGD
SCHEMBL11264404 0.76 ALDH1A1 (0.45) GAAGLO1LMNAKMT2AALDH1A1
SCHEMBL11256199 0.75 GAA (0.47) GAAGLO1LMNAKMT2AALDH1A1
SCHEMBL11385493 0.75 GAA (0.47) GAAGLO1LMNAKMT2AALDH1A1
SCHEMBL11257484 0.74 ALDH1A1 (0.45) GAAGLO1LMNAKMT2AALDH1A1
SCHEMBL11267322 0.73 SMN1; SMN2 (0.43) LMNAKMT2AALDH1A1CYP3A4CYP2C9
SCHEMBL13916496 0.71 CYP2C19 (0.52) GAALMNAKMT2AALDH1A1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0212340-B1 2-(heteroalkyl)-1,4-dihydropyridines, process for their preparations and pharmaceutical compositions containing them BOEHRINGER MANNHEIM ITALIA (IT) 1993-10-27 EP disclosed
US-4839348-A HYPOTENSIVE AGENTS; ANTICOAGULANTS, ANTIISCHEMIC AGENTS BOEHRINGER BIOCHEMIA ROBIN S.P.A. (IT) 1989-06-13 US disclosed
EP-0212340-A1 2-(heteroalkyl)-1,4-dihydropyridines, process for their preparations and pharmaceutical compositions containing them BOEHRINGER MANNHEIM ITALIA S.P.A. (IT) 1987-03-04 EP disclosed